A preliminary study of dopamine D2/3 receptor availability and social status in healthy and cocaine dependent humans imaged with [(11)C](+)PHNO

Drug Alcohol Depend. 2015 Sep 1:154:167-73. doi: 10.1016/j.drugalcdep.2015.06.039. Epub 2015 Jun 30.

Abstract

Background: Previous work in healthy non-human primates and humans has shown that social status correlates positively with dopamine 2/3 receptor (D2/3R) availability imaged with antagonist radioligands and positron emission tomography (PET). Further work in non-human primates suggests that this relationship is disrupted by chronic cocaine administration. This exploratory study examined the relationship between social status and D2/3R availability in healthy (HH) and cocaine dependent (CD) humans using the D3-preferring, agonist radioligand, [(11)C](+)PHNO.

Methods: Sixteen HH and sixteen CD individuals completed the Barratt Simplified Measure of Social Status (BSMSS) and underwent [(11)C](+)PHNO scanning to measure regional brain D2/3R binding potentials (BPND). Correlations between BPND and BSMSS scores were then assessed within each group.

Results: Within HH and CD groups, inverse associations between BSMSS score and BPND were observed in the substantia nigra/ventral tegmental area (SN/VTA) and the ventral striatum, and for the CD group alone, the amygdala. After adjusting for body mass index and age, negative correlations remained significant in the SN/VTA for HH and in the amygdala for CD subjects.

Conclusion: These preliminary data utilizing a dopamine agonist tracer demonstrate, for the first time, an inverse association between social status and D2/3R availability in the D3R rich extrastriatal regions of HH and CD humans.

Keywords: Cocaine; Dopamine; PET imaging; Social status; [(11)C](+)PHNO.

Publication types

  • Research Support, N.I.H., Extramural

MeSH terms

  • Adult
  • Amygdala / metabolism
  • Case-Control Studies
  • Cocaine-Related Disorders / metabolism*
  • Dopamine Agonists / metabolism*
  • Female
  • Functional Neuroimaging
  • Hierarchy, Social*
  • Humans
  • Male
  • Oxazines / metabolism*
  • Positron-Emission Tomography
  • Receptors, Dopamine D2 / metabolism*
  • Receptors, Dopamine D3 / metabolism*
  • Substantia Nigra / metabolism
  • Ventral Tegmental Area / metabolism
  • Young Adult

Substances

  • Dopamine Agonists
  • Oxazines
  • Receptors, Dopamine D2
  • Receptors, Dopamine D3
  • naxagolide