Anti-α4 Integrin Antibody Blocks Monocyte/Macrophage Traffic to the Heart and Decreases Cardiac Pathology in a SIV Infection Model of AIDS

J Am Heart Assoc. 2015 Jul 16;4(7):e001932. doi: 10.1161/JAHA.115.001932.

Abstract

Background: Cardiovascular disease (CVD), myocarditis and fibrosis are comorbidities of HIV(+) individuals on durable antiretroviral therapy (ART). Although mechanisms for these vary, monocytes/macrophages are increasingly demonstrated to be key players.

Methods and results: We directly blocked monocyte/macrophage traffic to the heart in an SIV model of AIDS using an anti-alpha-4 integrin antibody (natalizumab). Nineteen Rhesus macaques were SIVmac251 infected and CD8-lymphocyte depleted for the development of rapid AIDS. Ten animals received natalizumab once a week, for 3 weeks, and were sacrificed 1 week later. Six animals began treatment at the time of infection (early) and the remaining 4 began treatment 28 days post-infection (late), a time point we have previously established when significant cardiac inflammation occurs. Nine animals were untreated controls; of these, 3 were sacrificed early and 6 were sacrificed late. At necropsy, we found decreased SIV-associated cardiac pathology in late natalizumab-treated animals, compared to untreated controls. Early and late treatment resulted in significant reductions in numbers of CD163(+) and CD68(+) macrophages in cardiac tissues, compared to untreated controls, and a trend in decreasing numbers of newly recruited MAC387(+) and BrdU(+) (recruited) monocytes/macrophages. In late treated animals, decreased macrophage numbers in cardiac tissues correlated with decreased fibrosis. Early and late treatment resulted in decreased cardiomyocyte damage.

Conclusions: These data demonstrate a role for macrophages in the development of cardiac inflammation and fibrosis, and suggest that blocking monocyte/macrophage traffic to the heart can alleviate HIV- and SIV-associated myocarditis and fibrosis. They underscore the importance of targeting macrophage activation and traffic as an adjunctive therapy in HIV infection.

Keywords: HIV; animal model; cardiomyopathy; fibrosis; myocarditis.

Publication types

  • Research Support, N.I.H., Extramural

MeSH terms

  • Animals
  • Antigens, CD / metabolism
  • Antigens, Differentiation, Myelomonocytic / metabolism
  • CD8-Positive T-Lymphocytes / immunology
  • CD8-Positive T-Lymphocytes / virology
  • Cardiomyopathies / diagnosis
  • Cardiomyopathies / immunology
  • Cardiomyopathies / metabolism
  • Cardiomyopathies / prevention & control*
  • Cardiomyopathies / virology
  • Chemotaxis / drug effects*
  • Cytoprotection
  • Disease Models, Animal
  • Fibrosis
  • Immunocompromised Host
  • Immunologic Factors / pharmacology*
  • Integrin alpha4 / immunology*
  • Integrin alpha4 / metabolism
  • Macaca mulatta
  • Macrophages / drug effects*
  • Macrophages / immunology
  • Macrophages / metabolism
  • Macrophages / virology
  • Monocytes / drug effects*
  • Monocytes / immunology
  • Monocytes / metabolism
  • Monocytes / virology
  • Myocarditis / diagnosis
  • Myocarditis / immunology
  • Myocarditis / metabolism
  • Myocarditis / prevention & control*
  • Myocarditis / virology
  • Myocardium / immunology*
  • Myocardium / metabolism
  • Myocardium / pathology
  • Natalizumab / pharmacology*
  • Receptors, Cell Surface / metabolism
  • Simian Acquired Immunodeficiency Syndrome / diagnosis
  • Simian Acquired Immunodeficiency Syndrome / drug therapy*
  • Simian Acquired Immunodeficiency Syndrome / immunology
  • Simian Acquired Immunodeficiency Syndrome / metabolism
  • Simian Acquired Immunodeficiency Syndrome / virology
  • Simian Immunodeficiency Virus / immunology
  • Simian Immunodeficiency Virus / pathogenicity
  • Time Factors

Substances

  • Antigens, CD
  • Antigens, Differentiation, Myelomonocytic
  • CD163 antigen
  • Immunologic Factors
  • Natalizumab
  • Receptors, Cell Surface
  • Integrin alpha4