A liquid crystal of ascorbyl palmitate, used as vaccine platform, provides sustained release of antigen and has intrinsic pro-inflammatory and adjuvant activities which are dependent on MyD88 adaptor protein

J Control Release. 2015 Sep 28:214:12-22. doi: 10.1016/j.jconrel.2015.07.008. Epub 2015 Jul 15.

Abstract

Modern subunit vaccines require the development of new adjuvant strategies. Recently, we showed that CpG-ODN formulated with a liquid crystal nanostructure formed by self-assembly of 6-O-ascorbyl palmitate (Coa-ASC16) is an attractive system for promoting an antigen-specific immune response to weak antigens. Here, we showed that after subcutaneous injection of mice with near-infrared fluorescent dye-labeled OVA antigen formulated with Coa-ASC16, the dye-OVA was retained at the injection site for a longer period than when soluble dye-OVA was administered. Coa-ASC16 alone elicited a local inflammation, but how this material triggers this response has not been described yet. Although it is known that some materials used as a platform are not immunologically inert, very few studies have directly focused on this topic. In this study, we explored the underlying mechanisms concerning the interaction between Coa-ASC16 and the immune system and we found that the whole inflammatory response elicited by Coa-ASC16 (leukocyte recruitment and IL-1β, IL-6 and IL-12 production) was dependent on the MyD88 protein. TLR2, TLR4, TLR7 and NLRP3-inflammasome signaling were not required for induction of this inflammatory response. Coa-ASC16 induced local release of self-DNA, and in TLR9-deficient mice IL-6 production was absent. In addition, Coa-ASC16 revealed an intrinsic adjuvant activity which was affected by MyD88 and IL-6 absence. Taken together these results indicate that Coa-ASC16 used as a vaccine platform is effective due to the combination of the controlled release of antigen and its intrinsic pro-inflammatory activity. Understanding how Coa-ASC16 works might have significant implications for rational vaccine design.

Keywords: Ascorbyl palmitate; Controlled release; Danger-associated molecular patterns (DAMPs); Liquid crystal; Nanostructure; Vaccine adjuvant.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Adjuvants, Immunologic / chemistry*
  • Animals
  • Antigens / administration & dosage*
  • Ascorbic Acid / analogs & derivatives*
  • Ascorbic Acid / chemistry
  • Delayed-Action Preparations
  • Humans
  • Inflammasomes / drug effects
  • Inflammation / chemically induced
  • Inflammation / pathology
  • Interleukins / biosynthesis
  • Leukocytes / drug effects
  • Liquid Crystals
  • Mice
  • Mice, Knockout
  • Myeloid Differentiation Factor 88 / genetics
  • Myeloid Differentiation Factor 88 / metabolism*
  • Ovalbumin / immunology
  • Toll-Like Receptor 9 / biosynthesis
  • Toll-Like Receptor 9 / genetics
  • Toll-Like Receptors / biosynthesis
  • Vaccines / administration & dosage*

Substances

  • Adjuvants, Immunologic
  • Antigens
  • Delayed-Action Preparations
  • Inflammasomes
  • Interleukins
  • Myd88 protein, mouse
  • Myeloid Differentiation Factor 88
  • Tlr9 protein, mouse
  • Toll-Like Receptor 9
  • Toll-Like Receptors
  • Vaccines
  • Ovalbumin
  • Ascorbic Acid
  • 6-O-palmitoylascorbic acid