Erythromycin A oxime 11,12-carbonate and its oxime ethers

J Antibiot (Tokyo). 1989 Dec;42(12):1817-22. doi: 10.7164/antibiotics.42.1817.

Abstract

Erythromycin A oxime 11,12-carbonate (5a) and its oxime ethers 5b approximately 5p have been prepared and their antibacterial activities compared with those of erythromycin A (1) and its 11,12-carbonate 2. The oxime 5a and many of its oxime ether derivatives showed good activity in vitro against Gram-positive and the more permeable Gram-negative organisms, in some cases being even more active than the carbonate 2.

Publication types

  • Comparative Study

MeSH terms

  • Chemical Phenomena
  • Chemistry
  • Erythromycin / analogs & derivatives*
  • Erythromycin / chemical synthesis
  • Erythromycin / pharmacology
  • Ethers / chemical synthesis*
  • Ethers / pharmacology
  • Gram-Positive Bacteria / drug effects
  • Microbial Sensitivity Tests
  • Oximes / chemical synthesis*
  • Oximes / pharmacology

Substances

  • Ethers
  • Oximes
  • erythromycin A oxime 11,12-carbonate
  • Erythromycin