Sensitivity of glioma initiating cells to a monoclonal anti-EGFR antibody therapy under hypoxia

Life Sci. 2015 Sep 15:137:74-80. doi: 10.1016/j.lfs.2015.07.024. Epub 2015 Aug 1.

Abstract

Aims: Glioma initiating cells (GICs) represent a subpopulation of tumor cells endowed with self-renewal and multilineage differentiation capacity but also with innate resistance to cytotoxic agents, a feature likely to pose major clinical challenges towards the complete eradication of minimal residual disease in glioma patients.

Materials and methods: In this work, GICs were obtained from two patient-derived high-grade gliomas xenograft model, expressing differently EGFR. GICs were exposed to anti-EGFR monoclonal antibody cetuximab during 48h in 1% or 21% oxygen tension. Cell viability and self-renewal capacity were then evaluated as well as their angiogenic properties.

Key findings: GICs were sensitive to cetuximab only in normoxic condition whatever the EGFR status. Nevertheless, under hypoxia cetuximab was able to decrease the self-renewal capacity as well as the expression of CD133 while expression of GFAP increased. Moreover, cetuximab decreased the effect of GICs on endothelial cell migration under hypoxia.

Significance: Consequently, anti-EGFR therapy can be envisaged to target specifically GICs in order to limit the tumor recurrence.

Keywords: Angiogenesis; Anti-EGFR therapy; Glioma initiating cells; Hypoxia; Stemness.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Angiogenesis Modulating Agents / pharmacology
  • Antibodies, Monoclonal / immunology
  • Antibodies, Monoclonal / pharmacology
  • Antibodies, Monoclonal / therapeutic use*
  • Brain Neoplasms / drug therapy*
  • Brain Neoplasms / metabolism
  • Brain Neoplasms / pathology*
  • Cell Hypoxia*
  • Cell Movement
  • Cell Proliferation / drug effects
  • Cell Survival / drug effects
  • Cetuximab / pharmacology*
  • Endothelial Cells / drug effects
  • ErbB Receptors / antagonists & inhibitors*
  • ErbB Receptors / immunology
  • Gene Expression / drug effects
  • Glial Fibrillary Acidic Protein / metabolism
  • Glioma / drug therapy*
  • Glioma / metabolism
  • Glioma / pathology*
  • Humans
  • Neoplastic Stem Cells / drug effects*
  • Tumor Cells, Cultured

Substances

  • Angiogenesis Modulating Agents
  • Antibodies, Monoclonal
  • Glial Fibrillary Acidic Protein
  • EGFR protein, human
  • ErbB Receptors
  • Cetuximab