MYC and metabolism on the path to cancer

Semin Cell Dev Biol. 2015 Jul:43:11-21. doi: 10.1016/j.semcdb.2015.08.003. Epub 2015 Aug 12.

Abstract

The MYC proto-oncogene is frequently deregulated in human cancers, activating genetic programs that orchestrate biological processes to promote growth and proliferation. Altered metabolism characterized by heightened nutrients uptake, enhanced glycolysis and glutaminolysis and elevated fatty acid and nucleotide synthesis is the hallmark of MYC-driven cancer. Recent evidence strongly suggests that Myc-dependent metabolic reprogramming is critical for tumorigenesis, which could be attenuated by targeting specific metabolic pathways using small drug-like molecules. Understanding the complexity of MYC-mediated metabolic re-wiring in cancers as well as how MYC cooperates with other metabolic drivers such as mammalian target of rapamycin (mTOR) will provide translational opportunities for cancer therapy.

Keywords: Cancer; Metabolism; Myc; mTOR.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't
  • Review

MeSH terms

  • Cell Proliferation / physiology
  • Cell Transformation, Neoplastic / pathology*
  • Glucose / metabolism*
  • Glycolysis / physiology*
  • Homeostasis / physiology*
  • Humans
  • Neoplasms / pathology*
  • Proto-Oncogene Mas
  • Proto-Oncogene Proteins c-myc / genetics
  • Proto-Oncogene Proteins c-myc / metabolism*
  • TOR Serine-Threonine Kinases / metabolism
  • Transcriptional Activation / genetics

Substances

  • MAS1 protein, human
  • MYC protein, human
  • Proto-Oncogene Mas
  • Proto-Oncogene Proteins c-myc
  • MTOR protein, human
  • TOR Serine-Threonine Kinases
  • Glucose