Glioblastomas require integrin αvβ3/PAK4 signaling to escape senescence

Cancer Res. 2015 Nov 1;75(21):4466-73. doi: 10.1158/0008-5472.CAN-15-0988. Epub 2015 Aug 21.

Abstract

Integrin αvβ3 has been implicated as a driver of aggressive and metastatic disease, and is upregulated during glioblastoma progression. Here, we demonstrate that integrin αvβ3 allows glioblastoma cells to counteract senescence through a novel tissue-specific effector mechanism involving recruitment and activation of the cytoskeletal regulatory kinase PAK4. Mechanistically, targeting either αvβ3 or PAK4 led to emergence of a p21-dependent, p53-independent cell senescence phenotype. Notably, glioblastoma cells did not exhibit a similar requirement for either other integrins or additional PAK family members. Moreover, αvβ3/PAK4 dependence was not found to be critical in epithelial cancers. Taken together, our findings established that glioblastomas are selectively addicted to this pathway as a strategy to evade oncogene-induced senescence, with implications that inhibiting the αvβ3-PAK4 signaling axis may offer novel therapeutic opportunities to target this aggressive cancer.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Brain Neoplasms / genetics*
  • Brain Neoplasms / pathology
  • Cell Proliferation / genetics
  • Cellular Senescence / genetics*
  • Cyclin-Dependent Kinase Inhibitor p21 / genetics
  • Female
  • Glioblastoma / genetics*
  • Glioblastoma / pathology
  • Humans
  • Integrin alphaVbeta3 / genetics*
  • Integrin alphaVbeta3 / metabolism
  • Mice
  • Mice, Nude
  • Neoplasm Transplantation
  • RNA Interference
  • RNA, Small Interfering
  • Signal Transduction / genetics
  • Spheroids, Cellular
  • Transplantation, Heterologous
  • Tumor Cells, Cultured
  • Tumor Suppressor Protein p53 / genetics
  • Vitronectin / metabolism
  • p21-Activated Kinases / genetics*
  • p21-Activated Kinases / metabolism

Substances

  • Cyclin-Dependent Kinase Inhibitor p21
  • Integrin alphaVbeta3
  • RNA, Small Interfering
  • Tumor Suppressor Protein p53
  • Vitronectin
  • PAK4 protein, human
  • p21-Activated Kinases