Observational Retrospective Study of Altered Biodistribution of Tositumomab and 131I-Tositumomab

J Nucl Med. 2015 Nov;56(11):1800-3. doi: 10.2967/jnumed.115.156190. Epub 2015 Sep 3.

Abstract

The tositumomab/(131)I-tositumomab radioimmunotherapy regimen is administered as a dosimetric dose followed by a therapeutic dose. The biodistribution of the dosimetric dose is assessed by quantitative calculations of whole-body residence time (TBRT) and visual examination of whole-body γ-camera images, to determine the administered radioactivity dose and whether a therapeutic dose can be administered. We investigated whether altered biodistribution of (131)I-tositumomab could be identified using quantitative TBRT.

Methods: BioClinica, Inc., provided γ-camera images to an independent reviewer to assess altered (131)I-tositumomab biodistribution in patients reported to a registry.

Results: Of 2,649 therapeutic doses, 5 (0.2%) were cancelled because of altered biodistribution as determined by γ-camera images and TBRT. Of these, 3 γ-camera images were assessed by the independent reviewer; one showed altered biodistribution (0.04%) and was in agreement with the TBRT on-site calculation.

Conclusion: TBRT alone should be used to determine altered biodistribution and hence whether to administer the therapeutic dose.

Keywords: altered biodistribution; therapeutic dose; tositumomab.

Publication types

  • Observational Study
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Antibodies, Monoclonal / pharmacology*
  • Antineoplastic Agents / pharmacokinetics*
  • Antineoplastic Agents / therapeutic use
  • Dose-Response Relationship, Radiation
  • Humans
  • Iodine Radioisotopes
  • Lung / diagnostic imaging
  • Lung / metabolism
  • Lymphoma, Non-Hodgkin / diagnostic imaging
  • Lymphoma, Non-Hodgkin / drug therapy
  • Radionuclide Imaging
  • Retrospective Studies
  • Tissue Distribution
  • Whole Body Imaging

Substances

  • Antibodies, Monoclonal
  • Antineoplastic Agents
  • Iodine Radioisotopes
  • tositumomab I-131