Vitamin D prevents articular cartilage erosion by regulating collagen II turnover through TGF-β1 in ovariectomized rats

Osteoarthritis Cartilage. 2016 Feb;24(2):345-53. doi: 10.1016/j.joca.2015.08.013. Epub 2015 Sep 4.

Abstract

Objective: To explore the effect of vitamin D on turnover of articular cartilage with ovariectomy (OVX) induced OA, and to investigate transforming growth factor-β1 (TGF-β1) as a possible underlying mechanism mediated by 1α,25(OH)2D3.

Design: Sixty-six rats were randomly allocated into seven groups: sham plus control diet (SHAM+CTL), OVX+CTL diet, sham plus vitamin D-deficient (VDD) diet, OVX+VDD diet, and three groups of ovariectomized rats treated with different doses of 1α,25(OH)2D3. The cartilage erosion and the levels of serum 17β-estradiol, 1α,25(OH)2D3 and C-telopeptide of type II collagen (CTX-II) were measured. TGF-β1, type II Collagen (CII), matrix metalloproteinases (MMP)-9,-13 in articular cartilage were assessed by immunohistochemistry. TGF-β1 and CTX-II expression were measured in articular cartilage chondrocytes treated with/without tumor necrosis factor (TNF-α), 1α,25(OH)2D3, and TGF-β receptor inhibitor (SB505124) in vitro.

Results: Cartilage erosion due to OVX was significantly reduced in a dose-dependent manner by 1α,25(OH)2D3 supplementation, and exacerbated by VDD. The expressions of TGF-β1 and CII in articular cartilage were suppressed by OVX and VDD, and rescued by 1α,25(OH)2D3 supplementation. The expression of MMP-9,-13 in articular cartilage increased with OVX and VDD, and decreased with 1α,25(OH)2D3 supplementation. In vitro experiments showed that 1α,25(OH)2D3 increased the TGF-β1 expression of TNF-α stimulated chondrocytes in a dose-dependent manner. 1α,25(OH)2D3 significantly counteracted the increased CTX-II release due to TNF-α stimulation, and this effect was significantly suppressed by SB505124.

Conclusion: VDD aggravated cartilage erosion, and 1α,25(OH)2D3 supplementation showed protective effects in OVX-induced OA partly through the TGF-β1 pathway.

Keywords: Articular cartilage degradation; CTX-II; Chondrocytes; Ovariectomized rats; TGF-β1; Vitamin D.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Benzodioxoles / pharmacology
  • Calcitriol / blood
  • Calcitriol / pharmacology*
  • Cartilage, Articular / drug effects*
  • Cartilage, Articular / metabolism
  • Cartilage, Articular / pathology
  • Chondrocytes / drug effects*
  • Chondrocytes / metabolism
  • Collagen Type II / blood
  • Estradiol / blood
  • Female
  • Imidazoles / pharmacology
  • Immunohistochemistry
  • Ovariectomy*
  • Peptide Fragments / blood
  • Pyridines / pharmacology
  • Rats
  • Rats, Sprague-Dawley
  • Receptors, Transforming Growth Factor beta / antagonists & inhibitors
  • Transforming Growth Factor beta1 / drug effects*
  • Transforming Growth Factor beta1 / metabolism
  • Tumor Necrosis Factor-alpha / pharmacology
  • Vitamin D Deficiency / metabolism*
  • Vitamins / pharmacology*

Substances

  • 2-(5-benzo(1,3)dioxol-5-yl-2-tert-butyl-3H-imidazol-4-yl)-6-methylpyridine hydrochloride
  • Benzodioxoles
  • Collagen Type II
  • Imidazoles
  • Peptide Fragments
  • Pyridines
  • Receptors, Transforming Growth Factor beta
  • Tgfb1 protein, rat
  • Transforming Growth Factor beta1
  • Tumor Necrosis Factor-alpha
  • Vitamins
  • Estradiol
  • Calcitriol