Loganin protects against pancreatitis by inhibiting NF-κB activation

Eur J Pharmacol. 2015 Oct 15:765:541-50. doi: 10.1016/j.ejphar.2015.09.019. Epub 2015 Sep 25.

Abstract

Acute pancreatitis (AP) is an inflammatory disease of the pancreas, which, in its most severe form, is associated with multi-organ failure and death. Loganin, a major iridoid glycoside obtained from Corni fructus, has been shown to have anti-inflammatory and anti-shock effects. However, the effects of loganin on AP have not been determined. Pre-treatment of loganin reduced pancreatic damage and AP-associated lung injury and attenuated the severity of AP, as evidenced by (1) a reduction in several biochemical parameters (pancreatic weight to body weight ratio, myeloperoxidase activity, and level of amylase) and (2) production of pro-inflammatory cytokines such as interleukin (IL)-1β and tumor necrosis factor (TNF)-α. However, post-treatment of loganin failed to improve pancreatic damage and biochemical parameters of AP, but could inhibit the AP-induced elevation of IL-1β and TNF-α significantly. In addition, cerulein-induced activation of nuclear factor (NF)-κB was inhibited in the pancreas by administration of loganin. In conclusion, these results suggest that loganin exhibits an anti-inflammatory effect in cases of AP and its pulmonary complications through inhibition of NF-κB activation.

Keywords: Acute pancreatitis; Loganin; Nuclear factor-κB; Proinflammatory cytokines.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Anti-Inflammatory Agents / pharmacology
  • Anti-Inflammatory Agents / therapeutic use
  • Dose-Response Relationship, Drug
  • Female
  • Iridoids / pharmacology
  • Iridoids / therapeutic use*
  • Mice
  • Mice, Inbred C57BL
  • NF-kappa B / antagonists & inhibitors*
  • NF-kappa B / metabolism*
  • Pancreatitis / metabolism*
  • Pancreatitis / prevention & control*
  • Protective Agents / pharmacology
  • Protective Agents / therapeutic use

Substances

  • Anti-Inflammatory Agents
  • Iridoids
  • NF-kappa B
  • Protective Agents
  • loganin