Importance of Adult Dmbx1 in Long-Lasting Orexigenic Effect of Agouti-Related Peptide

Endocrinology. 2016 Jan;157(1):245-57. doi: 10.1210/en.2015-1560. Epub 2015 Oct 27.

Abstract

Dmbx1 is a brain-specific homeodomain transcription factor expressed primarily during embryogenesis, and its systemic disruption (Dmbx1(-/-)) in the ICR mouse strain resulted in leanness associated with impaired long-lasting orexigenic effect of agouti-related peptide (AgRP). Because spatial and temporal expression patterns of Dmbx1 change dramatically during embryogenesis, it remains unknown when and where Dmbx1 plays a critical role in energy homeostasis. In the present study, the physiological roles of Dmbx1 were examined by its conditional disruption (Dmbx1(loxP/loxP)) in the C57BL/6 mouse strain. Although Dmbx1 disruption in fetal brain resulted in neonatal lethality, its disruption by synapsin promoter-driven Cre recombinase, which eliminated Dmbx1 expression postnatally, exempted the mice (Syn-Cre;Dmbx1(loxP/loxP) mice) from lethality. Syn-Cre;Dmbx1(loxP/loxP) mice show mild leanness and impaired long-lasting orexigenic action of AgRP, demonstrating the physiological relevance of Dmbx1 in the adult. Visualization of Dmbx1-expressing neurons in adult brain using the mice harboring tamoxifen-inducible Cre recombinase in the Dmbx1 locus (Dmbx1(CreERT2/+) mice) revealed Dmbx1 expression in small numbers of neurons in restricted regions, including the lateral parabrachial nucleus (LPB). Notably, c-Fos expression in LPB was increased at 48 hours after AgRP administration in Dmbx1(loxP/loxP) mice but not in Syn-Cre;Dmbx1(loxP/loxP) mice. These c-Fos-positive neurons in LPB did not coincide with neurons expressing Dmbx1 or melanocortin 4 receptor but did coincide with those expressing calcitonin gene-related peptide. Accordingly, Dmbx1 in the adult LPB is required for the long-lasting orexigenic effect of AgRP via the neural circuitry involving calcitonin gene-related peptide neurons.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Agouti-Related Protein / metabolism*
  • Agouti-Related Protein / pharmacology
  • Animals
  • Appetite Depressants / pharmacology
  • Appetite Regulation* / drug effects
  • Biomarkers / metabolism
  • Brain / cytology
  • Brain / drug effects
  • Brain / growth & development
  • Brain / metabolism
  • Crosses, Genetic
  • Gene Expression Regulation, Developmental* / drug effects
  • Genes, Reporter / drug effects
  • Genetic Loci / drug effects
  • Male
  • Mice, Inbred C57BL
  • Mice, Inbred ICR
  • Mice, Knockout
  • Mice, Transgenic
  • Nerve Tissue Proteins / genetics
  • Nerve Tissue Proteins / metabolism*
  • Neurons / cytology
  • Neurons / drug effects
  • Neurons / metabolism*
  • Otx Transcription Factors / genetics
  • Otx Transcription Factors / metabolism*
  • Parabrachial Nucleus / cytology
  • Parabrachial Nucleus / drug effects
  • Parabrachial Nucleus / growth & development
  • Parabrachial Nucleus / metabolism*
  • Peptide Fragments / pharmacology
  • Promoter Regions, Genetic / drug effects
  • Proto-Oncogene Proteins c-fos / metabolism
  • Tamoxifen / pharmacology

Substances

  • Agouti-Related Protein
  • Agrp protein, mouse
  • Appetite Depressants
  • Biomarkers
  • Nerve Tissue Proteins
  • Otx Transcription Factors
  • Otx3 protein, mouse
  • Peptide Fragments
  • Proto-Oncogene Proteins c-fos
  • agouti-related protein (86-132), human
  • Tamoxifen