Inhibition of streptozocin-induced insulitis and diabetes with lobenzarit in CD-1 mice

Diabetes. 1989 May;38(5):558-61. doi: 10.2337/diab.38.5.558.

Abstract

When multiple low doses (30 mg/kg body wt) of streptozocin were given to CD-1 mice, diabetes associated with L3T4 T-lymphocyte- and B-lymphocyte-predominant insulitis occurred. Thus, a model of type I (insulin-dependent) diabetes was obtained. To treat these diabetic mice, we administered lobenzarit (CCA), a newly synthesized immunomodulator. CCA (2 or 10 mg/kg body wt) significantly inhibited the progression of diabetes by suppressing the severity and incidence of insulitis. Insulin contents of the pancreas were preserved. The possibility that autoimmune-related diabetes can be treated with CCA warrants further attention.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Blood Glucose / analysis
  • Diabetes Mellitus, Experimental / drug therapy*
  • Hyperglycemia / drug therapy
  • Islets of Langerhans / drug effects*
  • Male
  • Mice
  • Mice, Inbred Strains
  • ortho-Aminobenzoates / therapeutic use*

Substances

  • Blood Glucose
  • ortho-Aminobenzoates
  • lobenzarit