Wittig Reaction: Domino Olefination and Stereoselectivity DFT Study. Synthesis of the Miharamycins' Bicyclic Sugar Moiety

Org Lett. 2015 Nov 20;17(22):5622-5. doi: 10.1021/acs.orglett.5b02849. Epub 2015 Nov 9.

Abstract

2-O-Acyl protected-d-ribo-3-uloses reacted with [(ethoxycarbonyl)methylene]triphenylphosphorane in acetonitrile to afford regio- and stereoselectively 2-(Z)-alkenes in 10-60 min under microwave irradiation. This domino reaction is proposed to proceed via tautomerization of 3-ulose to enol, acyl migration, tautomerization to the 3-O-acyl-2-ulose, and Wittig reaction. Alternatively, in chloroform, regioselective 3-olefination of 2-O-pivaloyl-3-uloses gave (E)-alkenes, key precursors for the miharamycins' bicyclic sugar moiety.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Alkenes / chemical synthesis*
  • Alkenes / chemistry
  • Carbohydrates / chemical synthesis*
  • Carbohydrates / chemistry
  • Combinatorial Chemistry Techniques
  • Molecular Structure
  • Nucleosides / chemical synthesis*
  • Nucleosides / chemistry*
  • Stereoisomerism

Substances

  • Alkenes
  • Carbohydrates
  • Nucleosides
  • miharamycin A
  • miharamycin B