Dexamethasone Disodium Phosphate Penetration Into the Human Aqueous Humor After Topical Application

Curr Eye Res. 2016 Jul;41(7):897-9. doi: 10.3109/02713683.2015.1083589. Epub 2015 Nov 18.

Abstract

Purpose: To study the amount of steroids that is found in the aqueous humor after topical administration of dexamethasone solution eye-drops and dexamethasone suspension eye-drops.

Materials and methods: One hundred seventeen consecutive patients of both genders 18 years or older, candidates for cataract surgery were randomly assigned to one of three groups. Fifty-one patients (group A) received a single instillation of a suspension containing tobramicin 0.3% mg/ml + dexamethasone 0.1% mg/ml; 56 patients (group B) received a single instillation of a solution containing tobramicin 0.3% mg/ml + dexamethasone 0.1% mg/ml; 10 patients (group C), control group, did not receive any drops. Samples were taken immediately before surgery from the anterior chamber and dexamethasone levels were measured using gas chromatography/mass spectrometry.

Results: The mean dexamethasone concentrations were 0.56 μM (min 0.00, max 3.25) in group A and 0.15 μM (min 0.00, max 2.93) in group B. Dexamethasone was not detected in samples from group C.

Conclusions: Dexamethasone suspension gives concentrations of steroids in the aqueous humor approximately three times higher than with dexamethasone solution drops.

Keywords: Aqueous humor; concentration; dexamethasone; solution; suspension.

Publication types

  • Randomized Controlled Trial

MeSH terms

  • Aged
  • Aqueous Humor / metabolism*
  • Cataract Extraction
  • Chromatography, High Pressure Liquid
  • Dexamethasone / administration & dosage
  • Dexamethasone / analogs & derivatives*
  • Dexamethasone / pharmacokinetics
  • Female
  • Glucocorticoids / administration & dosage
  • Glucocorticoids / pharmacokinetics
  • Humans
  • Male
  • Middle Aged
  • Ophthalmic Solutions / administration & dosage
  • Ophthalmic Solutions / pharmacokinetics
  • Postoperative Complications / prevention & control

Substances

  • Glucocorticoids
  • Ophthalmic Solutions
  • dexamethasone 21-phosphate
  • Dexamethasone