Induction of angiotensin-converting enzyme inhibitory activity by acid-limited proteolysis of glyceraldehyde 3-phosphate dehydrogenase

Biochem Biophys Res Commun. 1989 Jun 15;161(2):456-60. doi: 10.1016/0006-291x(89)92620-x.

Abstract

Angiotensin-converting enzyme (ACE) inhibitors were excised from glyceraldehyde 3-phosphate dehydrogenase (GAPDH) preparations of tuna and porcine muscles by heating at 120 degrees C for 5 min in 1 M AcOH-20 mM HCl. The inhibitors were then purified by successive chromatographies. The final product from tuna was identified as Pro-Thr-His-Ile-Lys-Trp-Gly-Asp, which was the ACE inhibitor obtained from tuna muscle [Kohama et al. (1988) Biochem. Biophys. Res. Commun. 155, 332-337]. The porcine ACE inhibitor was found to be Pro-Ala-Asn-Ile-Lys-Trp-Gly-Asp, which was identical to the porcine muscle GAPDH peptide 79-86. These results strongly suggested that the ACE inhibitory octapeptides derived from GAPDH proteins by acid-limited proteolysis at Asp-Pro and Asp-Ala peptide bonds.

MeSH terms

  • Amino Acid Sequence
  • Angiotensin-Converting Enzyme Inhibitors / biosynthesis*
  • Angiotensin-Converting Enzyme Inhibitors / isolation & purification
  • Animals
  • Glyceraldehyde-3-Phosphate Dehydrogenases / metabolism*
  • Kinetics
  • Molecular Sequence Data
  • Peptide Fragments / isolation & purification
  • Peptide Fragments / pharmacology*
  • Peptide Hydrolases / pharmacology
  • Swine
  • Tuna

Substances

  • Angiotensin-Converting Enzyme Inhibitors
  • Peptide Fragments
  • Glyceraldehyde-3-Phosphate Dehydrogenases
  • Peptide Hydrolases