Optimizing outcomes in clozapine rechallenge following neutropenia: a cohort analysis

J Clin Psychiatry. 2015 Nov;76(11):e1410-6. doi: 10.4088/JCP.14m09326.

Abstract

Objective: Certain patients with treatment-refractory schizophrenia may be rechallenged with clozapine following previous neutropenia. Evidence guiding patient selection and the effectiveness of lithium and granulocyte-colony stimulating factor (G-CSF) in rechallenge is limited, and factors associated with successful outcomes are unclear.

Method: Outcomes were studied in patients rechallenged with clozapine at a tertiary referral center between January 2007 and December 2013, following 1 or more previous trials terminated due to neutropenia, defined as an absolute neutrophil count (ANC) < 1.5 × 10(9)/L. Demographic characteristics, details of each clozapine trial including ANC, and coprescribed medication were extracted, and factors associated with rechallenge outcomes were examined.

Results: Nineteen patients underwent clozapine rechallenge following previous neutropenia; 4 (21%) experienced further neutropenia, 2 of which developed agranulocytosis. Compared to successfully rechallenged patients, unsuccessfully rechallenged patients were significantly older (t = 2.10, P = .05), experienced onset of neutropenia sooner (W = 10.0, P = .03), and were more commonly coprescribed valproate. In addition to 5 patients with benign ethnic neutropenia (BEN), 8 patients not of an ethnicity associated with BEN also had idiopathic low neutrophil counts at baseline; lithium and G-CSF coprescription facilitated successful rechallenge in these patients.

Conclusions: In this selected population, the initial neutropenia was unlikely to be related to clozapine in a substantial proportion of cases. This group was successfully rechallenged following careful consideration of the risks and benefits, and lithium and G-CSF contributed to allowing continued clozapine therapy. In addition to black patients, other ethnic groups can have persistently low ANC unrelated to clozapine.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Adult
  • Antimanic Agents / therapeutic use
  • Antipsychotic Agents / administration & dosage
  • Antipsychotic Agents / adverse effects
  • Antipsychotic Agents / pharmacology*
  • Clozapine / administration & dosage
  • Clozapine / adverse effects
  • Clozapine / pharmacology*
  • Cohort Studies
  • Drug Therapy, Combination
  • Female
  • Granulocyte Colony-Stimulating Factor / therapeutic use
  • Humans
  • Leukocyte Count
  • Lithium Compounds / therapeutic use
  • Male
  • Middle Aged
  • Neutropenia* / blood
  • Neutropenia* / chemically induced
  • Neutropenia* / ethnology
  • Neutrophils*
  • Outcome Assessment, Health Care*
  • Schizophrenia / blood
  • Schizophrenia / drug therapy*
  • Valproic Acid / therapeutic use
  • Young Adult

Substances

  • Antimanic Agents
  • Antipsychotic Agents
  • Lithium Compounds
  • Granulocyte Colony-Stimulating Factor
  • Valproic Acid
  • Clozapine