Grancalcin (GCA) modulates Toll-like receptor 9 (TLR9) mediated signaling through its direct interaction with TLR9

Eur J Immunol. 2016 Mar;46(3):712-24. doi: 10.1002/eji.201545567. Epub 2016 Jan 12.

Abstract

Toll-like receptors (TLRs) are playing important roles in stimulating the innate immune response and intensifying adaptive immune response against invading pathogens. Appropriate regulation of TLR activation is important to maintain a balance between preventing tumor activation and inhibiting autoimmunity. Toll-like receptor 9 (TLR9) senses microbial DNA in the endosomes of plasmacytoid dendritic cells and triggers myeloid differentiation primary response gene 88 (MyD88) dependent nuclear factor kappa B (NF-κB) pathways and type I interferon (IFN) responses. However, mechanisms of how TLR9 signals are mediated and which molecules are involved in controlling TLR9 functions remain poorly understood. Here, we report that penta EF-hand protein grancalcin (GCA) interacts and binds with TLR9 in a yeast two-hybrid system and an overexpression system. Using siRNA-mediated knockdown experiments, we also revealed that GCA positively regulates type I IFN production, cytokine/chemokine production through nuclear localization of interferon regulatory factor 7 (IRF7), NF-κB activation, and mitogen-activated protein kinase (MAPK) activation in plasmacytoid dendritic cells. Our results indicate that heterodimerization of GCA and TLR9 is important for TLR9-mediated downstream signaling and might serve to fine tune processes against viral infection.

Keywords: Grancalcin; IRF7; Plasmacytoid dendritic cells; TLR9 signaling; Type I interferon.

Publication types

  • Research Support, N.I.H., Extramural

MeSH terms

  • Calcium-Binding Proteins / immunology
  • Calcium-Binding Proteins / metabolism*
  • Cytokines / genetics
  • Dendritic Cells / immunology
  • Dendritic Cells / metabolism
  • Gene Knockdown Techniques
  • Humans
  • Interferon Regulatory Factor-7 / genetics
  • Interferon Type I / genetics
  • Mitogen-Activated Protein Kinases / metabolism
  • NF-kappa B / metabolism
  • RNA, Small Interfering / genetics
  • Signal Transduction*
  • Toll-Like Receptor 9 / genetics
  • Toll-Like Receptor 9 / immunology
  • Toll-Like Receptor 9 / metabolism*
  • Two-Hybrid System Techniques

Substances

  • Calcium-Binding Proteins
  • Cytokines
  • GCA protein, human
  • Interferon Regulatory Factor-7
  • Interferon Type I
  • NF-kappa B
  • RNA, Small Interfering
  • TLR9 protein, human
  • Toll-Like Receptor 9
  • Mitogen-Activated Protein Kinases