Synthetic antibiofilm peptides

Biochim Biophys Acta. 2016 May;1858(5):1061-9. doi: 10.1016/j.bbamem.2015.12.015. Epub 2015 Dec 23.

Abstract

Bacteria predominantly exist as multicellular aggregates known as biofilms that are associated with at least two thirds of all infections and exhibit increased adaptive resistance to conventional antibiotic therapies. Therefore, biofilms are major contributors to the global health problem of antibiotic resistance, and novel approaches to counter them are urgently needed. Small molecules of the innate immune system called host defense peptides (HDPs) have emerged as promising templates for the design of potent, broad-spectrum antibiofilm agents. Here, we review recent developments in the new field of synthetic antibiofilm peptides, including mechanistic insights, synergistic interactions with available antibiotics, and their potential as novel antimicrobials against persistent infections caused by biofilms. This article is part of a Special Issue entitled: Antimicrobial peptides edited by Karl Lohner and Kai Hilpert.

Keywords: Antibiotic resistance; Biofilms; Biomaterials; Persistent infections; Synergy; Synthetic peptides.

Publication types

  • Research Support, Non-U.S. Gov't
  • Review

MeSH terms

  • Animals
  • Antimicrobial Cationic Peptides / biosynthesis
  • Antimicrobial Cationic Peptides / chemical synthesis
  • Antimicrobial Cationic Peptides / pharmacology*
  • Bacterial Infections / drug therapy
  • Bacterial Infections / immunology
  • Bacterial Infections / microbiology
  • Biofilms / drug effects*
  • Biofilms / growth & development
  • Cell Membrane / chemistry
  • Cell Membrane / drug effects*
  • Cell Membrane / metabolism
  • Disease Models, Animal
  • Drug Design
  • Drug Resistance, Bacterial / drug effects
  • Drug Synergism
  • Gram-Negative Bacteria / chemistry
  • Gram-Negative Bacteria / drug effects*
  • Gram-Negative Bacteria / growth & development
  • Gram-Positive Bacteria / chemistry
  • Gram-Positive Bacteria / drug effects*
  • Gram-Positive Bacteria / growth & development
  • Humans
  • Immunologic Factors / biosynthesis
  • Immunologic Factors / chemical synthesis
  • Immunologic Factors / pharmacology*
  • Microbial Sensitivity Tests
  • Structure-Activity Relationship

Substances

  • Antimicrobial Cationic Peptides
  • Immunologic Factors