Evidence for association of SNPs in ABCB1 and CBR3, but not RAC2, NCF4, SLC28A3 or TOP2B, with chronic cardiotoxicity in a cohort of breast cancer patients treated with anthracyclines

Pharmacogenomics. 2016 Feb;17(3):231-40. doi: 10.2217/pgs.15.162. Epub 2016 Jan 22.

Abstract

Aims: Validation of associations for SNPs in RAC2, NCF4 and SLC28A3, identification of a novel association with a TOP2B SNP and screening 23 SNPs putatively relevant to anthracycline-induced cardiotoxicity.

Patients & methods: A total of 166 breast cancer patients treated with doxorubicin underwent echocardiogram, including 19 cases with systolic dysfunction (ejection fraction <55%) and 147 controls. Four high priority SNPs were tested in the primary analysis, with appropriate statistical correction, and 23 additional SNPs were screened in an uncorrected secondary analysis.

Results: Previously reported associations for RAC2, NCF4 and SLC28A3 could not be validated and a novel association with TOP2B was not discovered in this cohort (all p > 0.05), likely due to inadequate power. Two SNPs were identified in the uncorrected secondary analysis including a protective SNP in ABCB1 (3435C>T, p = 0.049) and a risk allele in CBR3 (V244M, p = 0.012).

Conclusion: The associations reported in prior publications and those discovered in this secondary analysis require further replication in independent cohorts.

Keywords: ABCB1; CBR3; NCF4; RAC2; SLC28A3; TOP2B; anthracycline; cardiotoxicity; doxorubicin; pharmacogenetic; systolic dysfunction.

Publication types

  • Observational Study
  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't

MeSH terms

  • ATP Binding Cassette Transporter, Subfamily B / genetics
  • Alcohol Oxidoreductases / genetics*
  • Anthracyclines / adverse effects*
  • Antineoplastic Agents / adverse effects*
  • Breast Neoplasms / drug therapy*
  • Breast Neoplasms / genetics
  • Cardiotoxicity / genetics*
  • Case-Control Studies
  • Chronic Disease
  • Cross-Sectional Studies
  • DNA Topoisomerases, Type II / genetics
  • DNA-Binding Proteins / genetics
  • Female
  • Genetic Association Studies
  • Genetic Predisposition to Disease
  • Humans
  • Membrane Transport Proteins / genetics
  • NADPH Oxidases / genetics
  • Poly-ADP-Ribose Binding Proteins
  • Polymorphism, Single Nucleotide
  • RAC2 GTP-Binding Protein
  • rac GTP-Binding Proteins / genetics

Substances

  • ABCB1 protein, human
  • ATP Binding Cassette Transporter, Subfamily B
  • Anthracyclines
  • Antineoplastic Agents
  • DNA-Binding Proteins
  • Membrane Transport Proteins
  • Poly-ADP-Ribose Binding Proteins
  • cif nucleoside transporter
  • Alcohol Oxidoreductases
  • CBR3 protein, human
  • NADPH Oxidases
  • NCF4 protein, human
  • rac GTP-Binding Proteins
  • DNA Topoisomerases, Type II
  • TOP2B protein, human