Esterase mediated resistance in deltamethrin resistant reference tick colony of Rhipicephalus (Boophilus) microplus

Exp Appl Acarol. 2016 Jun;69(2):239-48. doi: 10.1007/s10493-016-0032-7. Epub 2016 Mar 15.

Abstract

Monitoring of acaricide resistance is considered as one of the important facets of integrated tick management. In an attempt of development of resistance monitoring indicators, in the present study two reference tick lines of Rhipicephalus (Boophilus) microplus maintained in the Entomology laboratory, Indian Veterinary Research Institute (IVRI), Izatnagar, India, were studied to determine the possible contributing factors involved in development of resistance to deltamethrin. Electrophoretic profiling of esterase enzymes detected high activities of EST-1 in reference resistant tick colony designated as IVRI-IV whereas it was not detectable in reference susceptible IVRI-I line of R. (B.) microplus. Esterases were further characterized as carboxylesterase or acetylcholinesterase based on inhibitor study using PMSF, eserine sulphate, malathion, TPP and copper sulphate. It was concluded that an acetylcholinesterase, EST-1, possibly plays an important role for development of deltamethrin resistance in IVRI-IV colony of R. (B.) microplus.

Keywords: Esterases; IVRI-IV tick colony; India; Resistance; Rhipicephalus (Boophilus) microplus.

MeSH terms

  • Acaricides / pharmacology*
  • Animals
  • Arthropod Proteins / metabolism*
  • Drug Resistance*
  • Esterases / metabolism*
  • India
  • Larva / drug effects
  • Larva / enzymology
  • Larva / growth & development
  • Larva / physiology
  • Nitriles / pharmacology*
  • Pyrethrins / pharmacology*
  • Rhipicephalus / drug effects*
  • Rhipicephalus / enzymology
  • Rhipicephalus / growth & development
  • Rhipicephalus / physiology

Substances

  • Acaricides
  • Arthropod Proteins
  • Nitriles
  • Pyrethrins
  • decamethrin
  • Esterases