Structural Mechanism of Allosteric Activity Regulation in a Ribonucleotide Reductase with Double ATP Cones

Structure. 2016 Jun 7;24(6):906-17. doi: 10.1016/j.str.2016.03.025. Epub 2016 Apr 28.

Abstract

Ribonucleotide reductases (RNRs) reduce ribonucleotides to deoxyribonucleotides. Their overall activity is stimulated by ATP and downregulated by dATP via a genetically mobile ATP cone domain mediating the formation of oligomeric complexes with varying quaternary structures. The crystal structure and solution X-ray scattering data of a novel dATP-induced homotetramer of the Pseudomonas aeruginosa class I RNR reveal the structural bases for its unique properties, namely one ATP cone that binds two dATP molecules and a second one that is non-functional, binding no nucleotides. Mutations in the observed tetramer interface ablate oligomerization and dATP-induced inhibition but not the ability to bind dATP. Sequence analysis shows that the novel type of ATP cone may be widespread in RNRs. The present study supports a scenario in which diverse mechanisms for allosteric activity regulation are gained and lost through acquisition and evolutionary erosion of different types of ATP cone.

MeSH terms

  • Adenosine Triphosphate / metabolism*
  • Allosteric Regulation
  • Bacterial Proteins / chemistry
  • Bacterial Proteins / genetics
  • Bacterial Proteins / metabolism
  • Binding Sites
  • Crystallography, X-Ray
  • Models, Molecular
  • Mutation
  • Protein Binding
  • Protein Conformation
  • Pseudomonas aeruginosa / chemistry
  • Pseudomonas aeruginosa / enzymology*
  • Pseudomonas aeruginosa / genetics
  • Ribonucleotide Reductases / chemistry*
  • Ribonucleotide Reductases / genetics
  • Ribonucleotide Reductases / metabolism*

Substances

  • Bacterial Proteins
  • Adenosine Triphosphate
  • Ribonucleotide Reductases