PDK1 Is a Regulator of Epidermal Differentiation that Activates and Organizes Asymmetric Cell Division

Cell Rep. 2016 May 24;15(8):1615-23. doi: 10.1016/j.celrep.2016.04.051. Epub 2016 May 12.

Abstract

Asymmetric cell division (ACD) in a perpendicular orientation promotes cell differentiation and organizes the stratified epithelium. However, the upstream cues regulating ACD have not been identified. Here, we report that phosphoinositide-dependent kinase 1 (PDK1) plays a critical role in establishing ACD in the epithelium. Production of phosphatidyl inositol triphosphate (PIP3) is localized to the apical side of basal cells. Asymmetric recruitment of atypical protein kinase C (aPKC) and partitioning defective (PAR) 3 is impaired in PDK1 conditional knockout (CKO) epidermis. PDK1(CKO) keratinocytes do not undergo calcium-induced activation of aPKC or IGF1-induced activation of AKT and fail to differentiate. PDK1(CKO) epidermis shows decreased expression of Notch, a downstream effector of ACD, and restoration of Notch rescues defective expression of differentiation-induced Notch targets in vitro. We therefore propose that PDK1 signaling regulates the basal-to-suprabasal switch in developing epidermis by acting as both an activator and organizer of ACD and the Notch-dependent differentiation program.

MeSH terms

  • 3-Phosphoinositide-Dependent Protein Kinases / metabolism*
  • Animals
  • Asymmetric Cell Division*
  • Calcium / pharmacology
  • Cell Differentiation*
  • Cells, Cultured
  • Embryo, Mammalian / cytology
  • Embryo, Mammalian / enzymology
  • Epidermal Cells*
  • Epidermis / enzymology*
  • Keratinocytes / cytology
  • Keratinocytes / drug effects
  • Keratinocytes / metabolism
  • Mice, Knockout
  • Phenotype
  • Phosphatidylinositols / metabolism
  • Phosphorylation / drug effects
  • Protein Kinase C
  • Receptors, Notch / metabolism
  • Signal Transduction

Substances

  • Phosphatidylinositols
  • Receptors, Notch
  • phosphoinositide 3-phosphate
  • 3-Phosphoinositide-Dependent Protein Kinases
  • PKC-3 protein
  • Protein Kinase C
  • Calcium