Increased GVHD-related mortality with broad-spectrum antibiotic use after allogeneic hematopoietic stem cell transplantation in human patients and mice

Sci Transl Med. 2016 May 18;8(339):339ra71. doi: 10.1126/scitranslmed.aaf2311.

Abstract

Intestinal bacteria may modulate the risk of infection and graft-versus-host disease (GVHD) after allogeneic hematopoietic stem cell transplantation (allo-HSCT). Allo-HSCT recipients often develop neutropenic fever, which is treated with antibiotics that may target anaerobic bacteria in the gut. We retrospectively examined 857 allo-HSCT recipients and found that treatment of neutropenic fever with imipenem-cilastatin and piperacillin-tazobactam antibiotics was associated with increased GVHD-related mortality at 5 years (21.5% for imipenem-cilastatin-treated patients versus 13.1% for untreated patients, P = 0.025; 19.8% for piperacillin-tazobactam-treated patients versus 11.9% for untreated patients, P = 0.007). However, two other antibiotics also used to treat neutropenic fever, aztreonam and cefepime, were not associated with GVHD-related mortality (P = 0.78 and P = 0.98, respectively). Analysis of stool specimens from allo-HSCT recipients showed that piperacillin-tazobactam administration was associated with perturbation of gut microbial composition. Studies in mice demonstrated aggravated GVHD mortality with imipenem-cilastatin or piperacillin-tazobactam compared to aztreonam (P < 0.01 and P < 0.05, respectively). We found pathological evidence for increased GVHD in the colon of imipenem-cilastatin-treated mice (P < 0.05), but no difference in the concentration of short-chain fatty acids or numbers of regulatory T cells. Notably, imipenem-cilastatin treatment of mice with GVHD led to loss of the protective mucus lining of the colon (P < 0.01) and the compromising of intestinal barrier function (P < 0.05). Sequencing of mouse stool specimens showed an increase in Akkermansia muciniphila (P < 0.001), a commensal bacterium with mucus-degrading capabilities, raising the possibility that mucus degradation may contribute to murine GVHD. We demonstrate an underappreciated risk for the treatment of allo-HSCT recipients with antibiotics that may exacerbate GVHD in the colon.

MeSH terms

  • Animals
  • Anti-Bacterial Agents
  • CD4-Positive T-Lymphocytes / metabolism
  • Cilastatin / therapeutic use
  • Cilastatin, Imipenem Drug Combination
  • Colon / microbiology
  • Drug Combinations
  • Feces / microbiology
  • Female
  • Flow Cytometry
  • Gastrointestinal Microbiome / drug effects
  • Graft vs Host Disease / etiology
  • Graft vs Host Disease / microbiology*
  • Graft vs Host Disease / mortality*
  • Hematopoietic Stem Cell Transplantation / adverse effects*
  • Humans
  • Imipenem / therapeutic use
  • Interleukin-23
  • Mice
  • Mice, Inbred C57BL
  • Penicillanic Acid / analogs & derivatives
  • Penicillanic Acid / therapeutic use
  • Phylogeny
  • Piperacillin / therapeutic use
  • Piperacillin, Tazobactam Drug Combination
  • Transplantation, Homologous / adverse effects*
  • Verrucomicrobia / classification
  • Verrucomicrobia / drug effects
  • Verrucomicrobia / genetics

Substances

  • Anti-Bacterial Agents
  • Drug Combinations
  • Interleukin-23
  • Cilastatin
  • Piperacillin, Tazobactam Drug Combination
  • Imipenem
  • Penicillanic Acid
  • Cilastatin, Imipenem Drug Combination
  • Piperacillin