Association of Pharmacological Treatments for Obesity With Weight Loss and Adverse Events: A Systematic Review and Meta-analysis

JAMA. 2016 Jun 14;315(22):2424-34. doi: 10.1001/jama.2016.7602.

Abstract

Importance: Five medications have been approved for the management of obesity, but data on comparative effectiveness are limited.

Objective: To compare weight loss and adverse events among drug treatments for obesity using a systematic review and network meta-analysis.

Data sources: MEDLINE, EMBASE, Web of Science, Scopus, and Cochrane Central from inception to March 23, 2016; clinical trial registries.

Study selection: Randomized clinical trials conducted among overweight and obese adults treated with US Food and Drug Administration-approved long-term weight loss agents (orlistat, lorcaserin, naltrexone-bupropion, phentermine-topiramate, or liraglutide) for at least 1 year compared with another active agent or placebo.

Data extraction and synthesis: Two investigators identified studies and independently abstracted data using a predefined protocol. A Bayesian network meta-analysis was performed and relative ranking of agents was assessed using surface under the cumulative ranking (SUCRA) probabilities. Quality of evidence was assessed using GRADE criteria.

Main outcomes and measures: Proportions of patients with at least 5% weight loss and at least 10% weight loss, magnitude of decrease in weight, and discontinuation of therapy because of adverse events at 1 year.

Results: Twenty-eight randomized clinical trials with 29 018 patients (median age, 46 years; 74% women; median baseline body weight, 100.5 kg; median baseline body mass index, 36.1) were included. A median 23% of placebo participants had at least 5% weight loss vs 75% of participants taking phentermine-topiramate (odds ratio [OR], 9.22; 95% credible interval [CrI], 6.63-12.85; SUCRA, 0.95), 63% of participants taking liraglutide (OR, 5.54; 95% CrI, 4.16-7.78; SUCRA, 0.83), 55% taking naltrexone-bupropion (OR, 3.96; 95% CrI, 3.03-5.11; SUCRA, 0.60), 49% taking lorcaserin (OR, 3.10; 95% CrI, 2.38-4.05; SUCRA, 0.39), and 44% taking orlistat (OR, 2.70; 95% CrI, 2.34-3.09; SUCRA, 0.22). All active agents were associated with significant excess weight loss compared with placebo at 1 year-phentermine-topiramate, 8.8 kg (95% CrI, -10.20 to -7.42 kg); liraglutide, 5.3 kg (95% CrI, -6.06 to -4.52 kg); naltrexone-bupropion, 5.0 kg (95% CrI, -5.94 to -3.96 kg); lorcaserin, 3.2 kg (95% CrI, -3.97 to -2.46 kg); and orlistat, 2.6 kg (95% CrI, -3.04 to -2.16 kg). Compared with placebo, liraglutide (OR, 2.95; 95% CrI, 2.11-4.23) and naltrexone-bupropion (OR, 2.64; 95% CrI, 2.10-3.35) were associated with the highest odds of adverse event-related treatment discontinuation. High attrition rates (30%-45% in all trials) were associated with lower confidence in estimates.

Conclusions and relevance: Among overweight or obese adults, orlistat, lorcaserin, naltrexone-bupropion, phentermine-topiramate, and liraglutide, compared with placebo, were each associated with achieving at least 5% weight loss at 52 weeks. Phentermine-topiramate and liraglutide were associated with the highest odds of achieving at least 5% weight loss.

Publication types

  • Meta-Analysis
  • Research Support, N.I.H., Extramural
  • Review
  • Systematic Review

MeSH terms

  • Anti-Obesity Agents / adverse effects*
  • Anti-Obesity Agents / therapeutic use
  • Bayes Theorem
  • Benzazepines / adverse effects
  • Benzazepines / therapeutic use
  • Drug Combinations
  • Female
  • Fructose / adverse effects
  • Fructose / analogs & derivatives
  • Fructose / therapeutic use
  • Humans
  • Lactones / adverse effects
  • Lactones / therapeutic use
  • Liraglutide / adverse effects
  • Liraglutide / therapeutic use
  • Male
  • Middle Aged
  • Naltrexone / adverse effects
  • Naltrexone / therapeutic use
  • Obesity / drug therapy*
  • Orlistat
  • Phentermine / adverse effects
  • Phentermine / therapeutic use
  • Randomized Controlled Trials as Topic
  • Topiramate
  • Weight Loss*

Substances

  • Anti-Obesity Agents
  • Benzazepines
  • Drug Combinations
  • Lactones
  • Topiramate
  • Fructose
  • Naltrexone
  • lorcaserin
  • Liraglutide
  • Orlistat
  • Phentermine