A Co-Drug of Butyric Acid Derived from Fermentation Metabolites of the Human Skin Microbiome Stimulates Adipogenic Differentiation of Adipose-Derived Stem Cells: Implications in Tissue Augmentation

J Invest Dermatol. 2017 Jan;137(1):46-56. doi: 10.1016/j.jid.2016.07.030. Epub 2016 Aug 4.

Abstract

We show that Staphylococcus epidermidis, a commensal bacterium in the human skin microbiome, produces short-chain fatty acids by glycerol fermentation that can induce adipogenesis. Although the antimicrobial and anti-inflammatory activities of short-chain fatty acids have been previously well characterized, little is known about the contribution of short-chain fatty acids to the adipogenic differentiation of adipose-derived stem cells (ADSCs). We show that ADSCs differentiated into adipocytes and accumulated lipids in the cytoplasm when cultured with butyric acid, a principal short-chain fatty acid in the fermentation metabolites of S. epidermidis. Additionally, a co-drug, butyric acid 2-(2-butyryloxyethoxy) ethyl ester (BA-DEG-BA), released active butyric acid when it was intradermally injected into mouse ears and induced ADSC differentiation, characterized by an increased expression of cytoplasmic lipids and perilipin A. The BA-DEG-BA-induced adipogenic differentiation was mediated via peroxisome proliferator-activated receptor gamma. Furthermore, intradermal injection of ADSCs along with BA-DEG-BA into mouse ears markedly enhanced the adipogenic differentiation of ADSCs, leading to dermal augmentation. Our study introduces BA-DEG-BA as an enhancer of ADSC adipogenesis and suggests an integral interaction between the human skin microbiome and ADSCs.

Publication types

  • Comparative Study
  • Research Support, N.I.H., Extramural

MeSH terms

  • Adipocytes / cytology
  • Adipocytes / physiology
  • Adipose Tissue / cytology*
  • Adipose Tissue / metabolism
  • Animals
  • Butyric Acid / pharmacology*
  • Cell Differentiation
  • Culture Media, Conditioned
  • Female
  • Humans
  • Mice
  • Mice, Knockout
  • Microbiota / drug effects*
  • Microbiota / physiology
  • Real-Time Polymerase Chain Reaction / methods
  • Skin / cytology
  • Skin / microbiology
  • Staphylococcus epidermidis / drug effects
  • Staphylococcus epidermidis / metabolism*
  • Stem Cells / cytology*

Substances

  • Culture Media, Conditioned
  • Butyric Acid