MicroRNA-34b/c inhibits aldosterone-induced vascular smooth muscle cell calcification via a SATB2/Runx2 pathway

Cell Tissue Res. 2016 Dec;366(3):733-746. doi: 10.1007/s00441-016-2469-8. Epub 2016 Aug 8.

Abstract

Increasing evidence shows that aldosterone and specific microRNAs (miRs) contribute to vascular smooth muscle cell (VSMC) calcification. In this study, we aim to explore the mechanistic links between miR-34b/c and aldosterone in VSMC calcification. VSMC calcification models were established both in vitro and in vivo. First, the levels of aldosterone, miR-34b/c and special AT-rich sequence-binding protein 2 (SATB2) were measured. Then, miR-34b/c mimics or inhibitors were transfected into VSMCs to evaluate the function of miR-34b/c. Luciferase reporter assays were used to demonstrate whether SATB2 was a direct target of miR-34b/c. Aldosterone and SATB2 were found to be markedly upregulated during VSMC calcification, whereas miR-34b/c expression was downregulated. Treatment with the mineralocorticoid receptor (MR) antagonist eplerenone inhibited VSMC calcification. In aldosterone-induced VSMC calcification, miR-34b/c levels were downregulated and SATB2 protein was upregulated. Furthermore, miR-34b/c overexpression alleviated aldosterone-induced VSMC calcification as well as inhibited the expression of SATB2 protein, whereas miR-34b/c inhibition markedly enhanced VSMC calcification and upregulated SATB2 protein. In addition, luciferase reporter assays showed that SATB2 is a direct target of miR-34b/c in VSMCs. Overexpression of SATB2 induced Runx2 overproduction and VSMC calcification. Therefore, miR-34b/c participates in aldosterone-induced VSMC calcification via a SATB2/Runx2 pathway. As miR-34b/c appears to be a negative regulator, it has potential as a therapeutic target of VSMC calcification.

Keywords: Aldosterone; SATB2; Vascular calcification; Vascular smooth muscle cell; miR-34b/c.

MeSH terms

  • 3' Untranslated Regions / genetics
  • Aldosterone / pharmacology*
  • Animals
  • Aorta / drug effects
  • Base Sequence
  • Core Binding Factor Alpha 1 Subunit / genetics
  • Core Binding Factor Alpha 1 Subunit / metabolism*
  • Gene Expression Regulation / drug effects
  • Glycerophosphates / pharmacology
  • Male
  • Matrix Attachment Region Binding Proteins / genetics
  • Matrix Attachment Region Binding Proteins / metabolism*
  • MicroRNAs / genetics
  • MicroRNAs / metabolism*
  • Muscle, Smooth, Vascular / pathology*
  • Myocytes, Smooth Muscle / drug effects
  • Myocytes, Smooth Muscle / metabolism
  • Myocytes, Smooth Muscle / pathology*
  • Osteoblasts / drug effects
  • Osteoblasts / metabolism
  • Rats, Sprague-Dawley
  • Receptors, Mineralocorticoid / metabolism
  • Signal Transduction / drug effects*
  • Transcription Factors / genetics
  • Transcription Factors / metabolism*
  • Uremia / complications
  • Uremia / genetics
  • Vascular Calcification / complications
  • Vascular Calcification / genetics*
  • Vascular Calcification / pathology

Substances

  • 3' Untranslated Regions
  • Core Binding Factor Alpha 1 Subunit
  • Glycerophosphates
  • MIRN34 microRNA, rat
  • Matrix Attachment Region Binding Proteins
  • MicroRNAs
  • Receptors, Mineralocorticoid
  • SATB2 protein, rat
  • Transcription Factors
  • Aldosterone
  • beta-glycerophosphoric acid