Biosynthesis of paf-acether. XIV. Paf-acether output in murine peritoneal macrophages is regulated by the level of acetylhydrolase

Biochem Biophys Res Commun. 1989 Jul 14;162(1):475-82. doi: 10.1016/0006-291x(89)92022-6.

Abstract

Paf-acether (paf) synthesis was previously shown to be impaired in 24 hr-adherent and Bacillus Calmette-Guérin-activated murine peritoneal macrophages as compared to resident macrophages. We report here that the induction of acetylhydrolase was responsible for the decreased paf output in 24 hr-adherent macrophages. The kinetic analysis of the enzymes derived from 2 hr-, 24 hr- and BCG-activated adherent macrophages and from plasma revealed that the Km for paf was similar whatever the source of the acetylhydrolase whereas the Vmax was five-fold increased in 24 hr-cultured macrophages. The acetylhydrolase activity was Ca2+-independent and was not inhibited by addition of alkyl-acyl (long chain)-glycero-phosphocholine suggesting that the enzyme was not a phospholipase A2.

MeSH terms

  • 1-Alkyl-2-acetylglycerophosphocholine Esterase
  • Animals
  • Cell Fractionation
  • Cells, Cultured
  • Macrophage Activation
  • Macrophages / enzymology*
  • Macrophages / metabolism
  • Mice
  • Peritoneal Cavity
  • Phospholipases / physiology*
  • Phospholipases A / blood
  • Phospholipases A / metabolism
  • Phospholipases A / physiology*
  • Phospholipases A2
  • Platelet Activating Factor / biosynthesis*
  • Platelet Activating Factor / metabolism

Substances

  • Platelet Activating Factor
  • Phospholipases
  • Phospholipases A
  • Phospholipases A2
  • 1-Alkyl-2-acetylglycerophosphocholine Esterase