Phase 2 study of low-dose clofarabine plus cytarabine for patients with higher-risk myelodysplastic syndrome who have relapsed or are refractory to hypomethylating agents

Cancer. 2017 Feb 15;123(4):629-637. doi: 10.1002/cncr.30383. Epub 2016 Oct 14.

Abstract

Background: The outcome of patients with higher-risk myelodysplastic syndromes (MDS) after hypomethylating agent (HMA) failure is poor. This study evaluated the safety and activity of a combination of low-dose clofarabine and cytarabine for these patients.

Methods: Seventy patients with higher-risk MDS who had no response, progressed, or relapsed after at least 4 cycles of HMA therapy were treated.

Results: The median age was 72 years. Thirty-nine percent of the patients had high-risk disease according to the International Prognostic Scoring System, and 50% of the patients had poor-risk cytogenetics. Twenty-three percent of the patients had therapy-related MDS. The median number of prior cycles of HMA was 6 (range, 4-45). The overall response rate was 44%. The 6-week mortality rate was 9%. Grade 3 and higher nonhematologic toxicities were rare, but infections occurred in 52% of the patients, and fever of unknown origin occurred in 33%. The median overall survival (OS) was 10 months (95% confidence interval, 1-37 months). Thirteen percent of the patients underwent allogeneic stem cell transplantation. The responding patients had a median OS of 22 months, whereas the nonresponding patients had a median OS of 4 months. A complex karyotype was associated with worse response rates and OS.

Conclusions: The combination of low-dose clofarabine and cytarabine is clinically active in these patients with few treatment options. Cancer 2017;123:629-637. © 2016 American Cancer Society.

Keywords: clofarabine; cytarabine; hypomethylating agents; myelodysplastic syndromes; treatment failure.

Publication types

  • Clinical Trial, Phase II

MeSH terms

  • Adenine Nucleotides / adverse effects*
  • Adult
  • Aged
  • Aged, 80 and over
  • Arabinonucleosides / adverse effects*
  • Clofarabine
  • Cytarabine / adverse effects*
  • DNA Methylation / drug effects
  • Disease-Free Survival
  • Female
  • Humans
  • Male
  • Middle Aged
  • Myelodysplastic Syndromes / chemically induced
  • Myelodysplastic Syndromes / drug therapy*
  • Myelodysplastic Syndromes / genetics
  • Myelodysplastic Syndromes / pathology
  • Neoplasm Proteins / genetics
  • Neoplasms / complications
  • Neoplasms / drug therapy*
  • Neoplasms / epidemiology
  • Neoplasms / pathology
  • Treatment Outcome

Substances

  • Adenine Nucleotides
  • Arabinonucleosides
  • Neoplasm Proteins
  • Cytarabine
  • Clofarabine