miR-127 promotes EMT and stem-like traits in lung cancer through a feed-forward regulatory loop

Oncogene. 2017 Mar 23;36(12):1631-1643. doi: 10.1038/onc.2016.332. Epub 2016 Nov 21.

Abstract

The coordination between cellular differentiation and the mesenchymal/stem transition is essential for both embryo development and neoplasia, suggesting a mechanistic link between these two major processes. In this work we show that miR-127, an embryo-expressing lung miRNA, was prominently induced in lung adenocarcinoma and correlated with poor prognosis. Elevated miR-127 level drove a pronounced shift from the epithelial to the mesenchymal phenotype in cancer cells, and this shift was associated with their acquisition of stem-like traits, increased resistance to the epidermal growth factor receptor inhibitor and tumor-propagating potential. In contrast, antagonizing miR-127 markedly reversed this malignant transition, compromised the stem-like properties and the in vivo tumorigenic capability of cancer cells. Importantly, a regulatory loop involving the inflammatory signals NF-κB, miR-127 and tumor necrosis factor alpha-induced protein 3 was uncovered as a self-reinforcing circuitry that ensured an aggressive transition in lung cancer. Thus, this work identifies a novel molecular mechanism linking stemness, malignancy and inflammation, opening a new avenue for cancer treatment.

MeSH terms

  • 3' Untranslated Regions
  • Adenocarcinoma / genetics
  • Adenocarcinoma / metabolism
  • Adenocarcinoma / pathology
  • Adenocarcinoma of Lung
  • Antineoplastic Agents / pharmacology
  • Cell Movement / genetics
  • Cell Transformation, Neoplastic / genetics
  • Cell Transformation, Neoplastic / metabolism
  • Drug Resistance, Neoplasm / genetics
  • Epithelial-Mesenchymal Transition / genetics*
  • Gefitinib
  • Gene Expression Regulation, Neoplastic
  • Humans
  • Lung Neoplasms / drug therapy
  • Lung Neoplasms / genetics*
  • Lung Neoplasms / metabolism
  • Lung Neoplasms / pathology
  • MicroRNAs / genetics*
  • Models, Biological
  • NF-kappa B / metabolism
  • Neoplastic Stem Cells / metabolism*
  • Quinazolines / pharmacology
  • RNA Interference
  • Signal Transduction*
  • Tumor Necrosis Factor alpha-Induced Protein 3 / genetics
  • Tumor Necrosis Factor alpha-Induced Protein 3 / metabolism

Substances

  • 3' Untranslated Regions
  • Antineoplastic Agents
  • MIRN127 microRNA, human
  • MicroRNAs
  • NF-kappa B
  • Quinazolines
  • Tumor Necrosis Factor alpha-Induced Protein 3
  • Gefitinib