MicroRNA-497 Induces Apoptosis and Suppresses Proliferation via the Bcl-2/Bax-Caspase9-Caspase3 Pathway and Cyclin D2 Protein in HUVECs

PLoS One. 2016 Dec 5;11(12):e0167052. doi: 10.1371/journal.pone.0167052. eCollection 2016.

Abstract

Introduction: MicroRNAs play crucial roles in various types of diseases. However, to date, no information about the role of miR-497 in the development of atherosclerosis has been reported. This study investigated the possible role of miR-497 in vascular endothelial cell injury during the early stage of atherosclerosis.

Materials and methods: The expression level of miR-497 in human umbilical vein endothelial cells (HUVECs) exposed to ox-LDL was detected using qRT-PCR. To perform gain of function and loss of function analyses, miR-497 mimics were transfected into HUVECs, and miR-497 inhibitors were transfected into HUVECs stimulated with ox-LDL. Flow cytometry was used to analyze cell cycle progression and apoptosis. EdU and CCK-8 assays were employed to detect DNA synthesis and cell proliferation, respectively. After bioinformatics prediction, a dual Luciferase Reporter assay was used to analyze the direct target genes of miR-497. The mRNA and protein levels of the target genes were detected using qRT-PCR and western blot analyses, respectively. Caspase-9/3 activity was analyzed to determine the mechanism of endothelial dysfunction.

Results: We showed that miR-497 was significantly upregulated in HUVECs stimulated with ox-LDL. Ectopic expression of miR-497 suppressed cell proliferation, induced apoptosis and increased the activity of caspase-9/3. After verification, Bcl2 and CCND2 were shown to be direct target genes of miR-497 in HUVECs. MiR-497 significantly suppressed cell proliferation by arresting the cell cycle through the CCND2 protein and induced apoptosis through the Bcl2/Bax-caspase9-caspase3 pathway.

Conclusion: Overall, our study shows that miR-497 might play a role in the development of atherosclerosis by inducing apoptosis and suppressing the proliferation of vascular endothelial cells. Therefore, miR-497 could be a potential therapeutic target for the treatment of atherosclerosis.

MeSH terms

  • Apoptosis / genetics*
  • Atherosclerosis / genetics
  • Caspase 3 / genetics*
  • Caspase 9 / genetics*
  • Cell Proliferation / genetics*
  • Cells, Cultured
  • Cyclin D2 / genetics*
  • Human Umbilical Vein Endothelial Cells
  • Humans
  • Lipoproteins, LDL / genetics
  • MicroRNAs / genetics*
  • Proto-Oncogene Proteins c-bcl-2 / genetics*
  • RNA, Messenger
  • bcl-2-Associated X Protein / genetics*

Substances

  • CCND2 protein, human
  • Cyclin D2
  • Lipoproteins, LDL
  • MIRN497 microRNA, human
  • MicroRNAs
  • Proto-Oncogene Proteins c-bcl-2
  • RNA, Messenger
  • bcl-2-Associated X Protein
  • oxidized low density lipoprotein
  • Caspase 3
  • Caspase 9

Grants and funding

The authors received no specific funding for this work.