Mixed effects of caffeic acid phenethyl ester (CAPE) on joint inflammation, bone loss and gastrointestinal inflammation in a murine model of collagen antibody-induced arthritis

Inflammopharmacology. 2017 Feb;25(1):55-68. doi: 10.1007/s10787-016-0306-z. Epub 2017 Jan 3.

Abstract

Objective: To investigate the effect of caffeic acid phenethyl ester (CAPE) on local and systemic inflammation and bone loss in collagen antibody-induced arthritis (CAIA) mice.

Methods: Four groups of mice (n = 8 per group) were allocated; control, CAPE (1 mg/kg), CAIA and CAIA + CAPE (1 mg/kg). Local inflammation and bone loss were evaluated using clinical paw scores, in vivo micro-computed tomography (micro-CT), histological assessment and tartrate-resistant acid phosphatase (TRAP) staining. Serum levels of C-reactive protein (CRP) and C-terminal telopeptide (CTX-1) were measured by ELISA. Jejunum and colon sections were evaluated histopathologically for damage and toxicity.

Results: Greater paw scores and percentage change in paw volume were observed in CAIA + CAPE compared to the control groups (p < 0.05). Bone volume over time remained unchanged (p = 0.94) and the number of multinucleated TRAP-positive cells was greatest in CAIA + CAPE mice (p < 0.05). CRP and CTX-1 levels did not differ between groups. CAIA + CAPE mice exhibited lower colon toxicity scores and a reduced percentage of cavitated goblet cells in the colon crypts compared with CAIA mice (p = 0.026 and p = 0.003, respectively). Histopathology in the jejunum was not altered.

Conclusion: CAPE did not reduce paw inflammation or bone loss in CAIA mice. CAPE reduced histopathological changes in the colon of CAIA mice.

Keywords: Bone; CAIA; CAPE; Gastrointestinal tract; Inflammatory arthritis; Micro-CT.

MeSH terms

  • Animals
  • Arthritis, Experimental / diagnostic imaging*
  • Arthritis, Experimental / drug therapy*
  • Bone Resorption / diagnostic imaging*
  • Bone Resorption / drug therapy*
  • Caffeic Acids / therapeutic use*
  • Collagen / toxicity
  • Gastrointestinal Tract / diagnostic imaging*
  • Gastrointestinal Tract / drug effects
  • Inflammation / chemically induced
  • Inflammation / diagnostic imaging
  • Inflammation / drug therapy
  • Joints / diagnostic imaging
  • Joints / drug effects
  • Mice
  • Mice, Inbred BALB C
  • Phenylethyl Alcohol / analogs & derivatives*
  • Phenylethyl Alcohol / therapeutic use
  • Random Allocation
  • Tomography, X-Ray Computed
  • Treatment Outcome

Substances

  • Caffeic Acids
  • Collagen
  • caffeic acid phenethyl ester
  • Phenylethyl Alcohol