[The effect of mucous excipient concentration on bioadhesion ex vivo]

Pharmazie. 1989 Jul;44(7):460-2.
[Article in German]

Abstract

The bioadhesion of aqueous solutions of polyacrylics (1-3), hydroxyethylcellulose (4), sodium carboxymethylamylopectin (5), polyvinylalcohol (6) and tragant (7) was investigated using a tensiometer and fresh intestine of pigs. It was dependent on the concentration of the excipient as described by a quadratic equation and found in the maximum from 244 Pa (7) to 554 Pa (4). The maximum of bioadhesion corresponds to the concentration of the excipient from 0.15% (2) to 23.7% (4) and to the viscosity of the solutions from 0.11 Pa.s (3) to 3.6.10(6) Pa.s (4). There was not a correlation between the viscosity and the bioadhesion.

Publication types

  • English Abstract

MeSH terms

  • Adhesiveness
  • Animals
  • Excipients
  • In Vitro Techniques
  • Intestinal Absorption*
  • Regression Analysis
  • Swine
  • Viscosity

Substances

  • Excipients