Impact of ITPA gene polymorphisms on the risk of ribavirin-induced haemolytic anaemia using interferon-free antivirals for chronic hepatitis C

Antivir Ther. 2017;22(7):571-575. doi: 10.3851/IMP3138. Epub 2017 Feb 15.

Abstract

Background: Single nucleotide polymorphisms (SNPs) at the ITPA gene are associated with haemolytic anaemia in chronic hepatitis C patients treated with pegylated interferon-ribavirin (RBV). Information in patients treated with interferon-free, direct-acting antivirals (DAA) is scarce.

Methods: Median haemoglobin (Hb) levels were compared at baseline and at week 4, when ribavirin concentration achieves steady state, in all consecutive chronic hepatitis C patients treated with oral DAA plus RBV at our clinic.

Results: Median Hb drop in 55 patients was greater in rs1127354-CC than -CA/AA (1.8 versus 0.7 g/dl; P=0.029), and in rs6051702-AA than -AC/CC carriers (2.2 versus 1.1 g/dl; P=0.016). Eleven (20%) patients experienced severe anaemia, defined as Hb drop >3 g/dl or to <10 g/dl. All of them were rs6051702-AA.

Conclusions: Baseline testing of rs6051702 may identify the subset of patients at greatest risk for RBV-induced anaemia using interferon-free hepatitis C therapies.

MeSH terms

  • Adult
  • Aged
  • Alleles
  • Anemia, Hemolytic / etiology*
  • Antiviral Agents / adverse effects*
  • Antiviral Agents / therapeutic use
  • Disease Susceptibility*
  • Female
  • Genotype
  • Hepatitis C, Chronic / complications*
  • Hepatitis C, Chronic / drug therapy
  • Humans
  • Male
  • Middle Aged
  • Polymorphism, Single Nucleotide*
  • Pyrophosphatases / genetics*
  • Retrospective Studies
  • Ribavirin / adverse effects*
  • Ribavirin / therapeutic use

Substances

  • Antiviral Agents
  • Ribavirin
  • Pyrophosphatases
  • ITPA protein, human