Characterization of erythropoietin receptor on erythropoietin-unresponsive mouse erythroleukemia cells

Biochim Biophys Acta. 1988 Aug 18;943(2):326-30. doi: 10.1016/0005-2736(88)90564-0.

Abstract

A membrane receptor for erythropoietin was identified in various erythropoietin-unresponsive mouse erythroleukemia cells. Scatchard analyses of the binding of human 125I-labeled erythropoietin to T3C1-2-0, K-1, GM86 and 707 cells showed the presence of a single class of binding sites with apparent Kd values of 0.27-0.78 nM, which are slightly higher than those of erythropoietin-responsive cells. The number of binding sites varied from 110 to 930 per cell. Crosslinking of 125I-erythropoietin to its binding sites with disuccinimidyl suberate revealed the existence of a single binding protein with molecular mass of 63 kDa. No binding sites with higher molecular mass, as observed in erythropoietin-responsive cells, were detected, nor was any specific binding observed to the non-erythroid hematopoietic cell or to the human erythroleukemia cells examined.

Publication types

  • Comparative Study

MeSH terms

  • Animals
  • Cross-Linking Reagents
  • Electrophoresis, Polyacrylamide Gel
  • Erythropoietin / metabolism*
  • Erythropoietin / pharmacology
  • Hematopoietic Stem Cells
  • Humans
  • Iodine Radioisotopes
  • Leukemia, Erythroblastic, Acute / metabolism*
  • Mice
  • Molecular Weight
  • Receptors, Cell Surface / metabolism*
  • Receptors, Erythropoietin
  • Recombinant Proteins / metabolism
  • Succinimides
  • Tumor Cells, Cultured

Substances

  • Cross-Linking Reagents
  • Iodine Radioisotopes
  • Receptors, Cell Surface
  • Receptors, Erythropoietin
  • Recombinant Proteins
  • Succinimides
  • Erythropoietin
  • disuccinimidyl suberate