What's in a side effect? The association between pulmonary vasodilator adverse drug events and clinical outcomes in patients with pulmonary arterial hypertension

Int J Cardiol. 2017 Aug 1:240:386-391. doi: 10.1016/j.ijcard.2017.04.016. Epub 2017 Apr 6.

Abstract

Background: Adverse drug events (ADEs) with pulmonary vasodilator use in pulmonary arterial hypertension (PAH) are common. ADEs may contribute to worse quality of life; however, their relationship to prognosis is unknown. The objective of this study was to determine whether common ADEs after initiating subcutaneous treprostinil were associated with prognosis in PAH.

Methods: We assembled a retrospective cohort of participants from four clinical trials of treprostinil for PAH, including 908 participants who received subcutaneous treprostinil and 243 who received placebo at the time ADEs were ascertained. The occurrences of four common early ADEs (infusion reactions, headaches, jaw pain, or gastrointestinal side effects) were assessed during the eight weeks after starting the infusion. We used Cox proportional hazards to estimate associations between ADEs and mortality.

Results: No ADEs related to placebo were associated with mortality. In participants who received treprostinil, infusion reactions, headaches, and jaw pain were not associated with mortality. Gastrointestinal side effects occurring during the first eight weeks following treprostinil infusion were associated with a 57% increase in the hazard of mortality (95% CI: 14-118%). This relationship was unchanged after adjusting for demographic differences and differences in baseline PAH severity.

Conclusions: Gastrointestinal ADEs after starting subcutaneous treprostinil were associated with an increased risk for mortality. Increased mortality was not observed with other early ADEs or with gastrointestinal symptoms in participants who were not receiving treprostinil at the time. This hypothesis-generating association suggests ADEs may identify different phenotypes in PAH.

Keywords: Epidemiology; Pulmonary hypertension; Side effects.

Publication types

  • Clinical Trial, Phase II
  • Clinical Trial, Phase III
  • Observational Study

MeSH terms

  • Adult
  • Antihypertensive Agents / adverse effects*
  • Cohort Studies
  • Drug-Related Side Effects and Adverse Reactions / etiology*
  • Drug-Related Side Effects and Adverse Reactions / mortality
  • Epoprostenol / adverse effects
  • Epoprostenol / analogs & derivatives*
  • Female
  • Gastrointestinal Diseases / chemically induced*
  • Gastrointestinal Diseases / mortality
  • Humans
  • Hypertension, Pulmonary / drug therapy*
  • Hypertension, Pulmonary / mortality
  • Male
  • Middle Aged
  • Retrospective Studies
  • Treatment Outcome
  • Vasodilator Agents / adverse effects*

Substances

  • Antihypertensive Agents
  • Vasodilator Agents
  • Epoprostenol
  • treprostinil