Elevated Plasma Aβ42 in Cognitively Impaired Individuals Taking ACE Inhibitor Antihypertensives

Am J Alzheimers Dis Other Demen. 2017 Sep;32(6):347-352. doi: 10.1177/1533317517707288. Epub 2017 Apr 27.

Abstract

Background/rationale: Accumulating evidence suggests that the use of angiotensin-converting enzyme inhibitor (ACE-I) medication protects against cognitive decline in the elderly patients. We investigated whether ACE-I use was associated with higher plasma levels of amyloid-β (Aβ), possibly indicating improved Aβ clearance from brain to blood.

Methods: We measured and compared plasma concentrations of Aβ42, Aβ40, and creatinine in cognitively impaired individuals with amnestic mild cognitive impairment, probable Alzheimer's disease (AD) dementia, and mixed probable AD/vascular dementia.

Results: Plasma Aβ42 levels and Aβ42/Aβ40 ratios of participants taking ACE-Is (n = 11) significantly exceeded ( t = 3.1, df = 19, P = .006; U = 24, P = .029, respectively) those not taking ACE-Is (n = 10).

Conclusions: This study is the first to show an association between ACE-I use and increased plasma Aβ42 level and Aβ42/Aβ40 ratio in cognitively impaired individuals. Future investigations should assess whether a possible ACE-I-induced increase in plasma Aβ42 indicates improved Aβ42 clearance from brain that contributes to protection from cognitive decline.

Keywords: Alzheimer’s disease; amyloid; angiotensin converting enzyme inhibitor; clearance; dementia; mild cognitive impairment.

MeSH terms

  • Aged
  • Aged, 80 and over
  • Alzheimer Disease / blood*
  • Amnesia / blood*
  • Amyloid beta-Peptides / blood*
  • Angiotensin-Converting Enzyme Inhibitors / pharmacology*
  • Cognitive Dysfunction / blood*
  • Creatine / blood
  • Dementia, Vascular / blood*
  • Female
  • Humans
  • Hypertension / drug therapy
  • Male
  • Peptide Fragments / blood*

Substances

  • Amyloid beta-Peptides
  • Angiotensin-Converting Enzyme Inhibitors
  • Peptide Fragments
  • amyloid beta-protein (1-40)
  • amyloid beta-protein (1-42)
  • Creatine