Heterologous up-regulation of the 1,25-dihydroxyvitamin D3 receptor by parathyroid hormone (PTH) and PTH-like peptide in osteoblast-like cells

Biochem Biophys Res Commun. 1988 Oct 14;156(1):588-94. doi: 10.1016/s0006-291x(88)80883-0.

Abstract

1,25-Dihydroxyvitamin D3 (1,25-(OH)2D3) receptor content in cultured osteogenic sarcoma cells (UMR-106) was found to be increased after treatment with both bovine and human PTH and human PTH-like peptide (hPLP). The dose dependent increase of receptors was preceded by a dose dependent stimulation of cAMP production. This suggests a role for cAMP as mediator of the PTH- and hPLP-induced 1,25-(OH)2D3 receptor up-regulation. Furthermore, evidence was obtained that new mRNA and de novo receptor synthesis is involved in this heterologous 1,25-(OH)2D3 receptor up-regulation.

MeSH terms

  • Animals
  • Calcitriol / metabolism*
  • Cell Line
  • Cyclic AMP / metabolism
  • Cycloheximide / pharmacology
  • Dactinomycin / pharmacology
  • Kinetics
  • Osteoblasts / metabolism
  • Osteosarcoma
  • Parathyroid Hormone / pharmacology*
  • Peptide Fragments / pharmacology*
  • Rats
  • Receptors, Calcitriol
  • Receptors, Steroid / biosynthesis
  • Receptors, Steroid / drug effects
  • Receptors, Steroid / metabolism*
  • Teriparatide

Substances

  • Parathyroid Hormone
  • Peptide Fragments
  • Receptors, Calcitriol
  • Receptors, Steroid
  • Teriparatide
  • Dactinomycin
  • Cycloheximide
  • Cyclic AMP
  • Calcitriol