Anti-androgenic effects of bisphenol-A on spatial memory and synaptic plasticity of the hippocampus in mice

Horm Behav. 2017 Jul:93:151-158. doi: 10.1016/j.yhbeh.2017.05.014. Epub 2017 Jun 9.

Abstract

Bisphenol-A (BPA) is a common environmental endocrine disruptor. Our recent studies found that exposure to BPA in both adolescent and adulthood sex-specifically impaired spatial memory in male mice. In this study, 11-week-old gonadectomied (GDX) male mice daily received subcutaneous injections of testosterone propionate (TP, 0.5mg/kg), TP and BPA (0.4 and 4mg/kg), or vehicle for 45days. The results of Morris water maze task showed that exposure to BPA did not affect the spatial memory of GDX mice but impaired that of sham (4mg/kg/day) and TP-treated GDX mice (0.4mg/kg/day). In addition, BPA reduced the level of testosterone (T) in the serum and brain of sham and TP-treated GDX mice. Exposure to BPA decreased the synaptic density and had an adverse effect on the synaptic interface of the hippocampus in sham and TP-treated GDX mice. The results of western blot analysis further showed that BPA (4mg/kg) reduced the levels of synaptic proteins (synapsin I and PSD-95) and NMDA receptor subunit NR2B in sham and TP-treated GDX mice. BPA decreased the phosphorylation of ERK1/2 but increased the phosphorylation of p38 in sham and TP-treated GDX mice. These results suggest that impairment of spatial memory and adverse effects on synaptic remodeling of hippocampal neurons in males after long-term BPA exposure is related to the anti-androgen effect of BPA. These effects of BPA may be associated with downregulated synaptic proteins and NMDA receptor through inhibiting ERKs and promoting the p38 pathways.

Keywords: Androgen; Bisphenol-A; Memory; Synaptic plasticity.

MeSH terms

  • Androgen Antagonists / pharmacology*
  • Animals
  • Benzhydryl Compounds / pharmacology*
  • Endocrine Disruptors / pharmacology*
  • Hippocampus / drug effects*
  • Hippocampus / metabolism
  • Hippocampus / physiology
  • Male
  • Mice
  • Mice, Inbred ICR
  • Neuronal Plasticity / drug effects*
  • Neurons / drug effects
  • Neurons / metabolism
  • Phenols / pharmacology*
  • Receptors, N-Methyl-D-Aspartate / metabolism
  • Spatial Memory / drug effects*
  • Synapsins / metabolism
  • Testosterone / metabolism

Substances

  • Androgen Antagonists
  • Benzhydryl Compounds
  • Endocrine Disruptors
  • NR2B NMDA receptor
  • Phenols
  • Receptors, N-Methyl-D-Aspartate
  • Synapsins
  • Testosterone
  • bisphenol A