Polymyxin B Attenuates LPS-Induced Death but Aggravates Radiation-Induced Death via TLR4-Myd88-IL-6 Pathway

Cell Physiol Biochem. 2017;42(3):1120-1126. doi: 10.1159/000478767. Epub 2017 Jun 29.

Abstract

Background/aims: Polymyxin B (PMB) is a cyclic cationic polypeptide antibiotic widely used to counteract the effects of endotoxin contamination, both in vitro and in vivo. Lipopolysaccharide (LPS) is an endotoxin that acts as a radiation protection factor. In this study, we focus on the role of PMB in LPS-induced and radiation-induced mortality in mice.

Methods: Mice received total-body radiation or were pretreated by LPS or PMB, and the survival of mice was recorded. Elisa were used to detect the cytokines levels.

Results: PMB decreased LPS-induced, but increased radiation-induced mortality in mice. Moreover, PMB could block the LPS-induced radioprotective effect. The ELISA and gene knock-out experiments indicated that PMB reduces TNF-α level to block LPS-induced mortality in mice, and inhibits IL-6, G-CSF and IL-10 to increase radiation-induced mortality via the TLR4-Myd88-IL-6 pathway.

Conclusions: Our study revealed a role of PMB in LPS-induced endotoxemia and radiation exposure. We infer that the TLR4-Myd88-IL-6 pathway may play a crucial role in the process.

Keywords: IL-6; LPS; Myd88; Polymyxin B; Radiation; TLR4.

MeSH terms

  • Animals
  • Anti-Bacterial Agents / pharmacology*
  • Granulocyte Colony-Stimulating Factor
  • Interleukin-6 / immunology*
  • Lipopolysaccharides / adverse effects*
  • Lipopolysaccharides / immunology
  • Mice
  • Myeloid Differentiation Factor 88 / immunology*
  • Polymyxin B / pharmacology*
  • Radiation Injuries / complications*
  • Radiation Injuries / mortality
  • Signal Transduction / drug effects
  • Signal Transduction / radiation effects
  • Toll-Like Receptor 4 / immunology*

Substances

  • Anti-Bacterial Agents
  • Interleukin-6
  • Lipopolysaccharides
  • Myd88 protein, mouse
  • Myeloid Differentiation Factor 88
  • Tlr4 protein, mouse
  • Toll-Like Receptor 4
  • Granulocyte Colony-Stimulating Factor
  • Polymyxin B