Therapeutic blockade of Foxp3 in experimental breast cancer models

Breast Cancer Res Treat. 2017 Nov;166(2):393-405. doi: 10.1007/s10549-017-4414-2. Epub 2017 Jul 29.

Abstract

Purpose: Regulatory T cells (Tregs) impair the clinical benefit of cancer immunotherapy. To optimize the antitumor efficacy of therapeutic dendritic cell (DC) vaccines, we aimed to inhibit Foxp3, a transcription factor required for Treg function.

Methods: Mice bearing established syngeneic LM3 and 4T1 breast tumors were treated with antitumor DC vaccines and a synthetic peptide (P60) that has been shown to inhibit Foxp3.

Results: Treatment with P60 improved the therapeutic efficacy of DC vaccines in these experimental models. In addition, monotherapy with P60 inhibited tumor growth in immunocompetent as well as in immuno-compromised animals bearing established tumors. We found expression of Foxp3 in human and murine breast tumor cells. P60 inhibited IL-10 secretion in breast cancer cells that expressed Foxp3.

Conclusions: Our results suggest that Foxp3 blockade improves the therapeutic efficacy of DC vaccines by inhibition of Tregs and through a direct antitumor effect. This strategy could prove useful to neutralize the immunosuppressive microenvironment and to boost antitumor immunity in breast cancer.

Keywords: Breast cancer; Dendritic cell vaccines; Foxp3; Immunotherapy; Regulatory T cells.

MeSH terms

  • Animals
  • Breast Neoplasms / immunology
  • Breast Neoplasms / metabolism
  • Breast Neoplasms / therapy*
  • Cancer Vaccines / administration & dosage
  • Cancer Vaccines / pharmacology
  • Cell Line, Tumor
  • Cell-Penetrating Peptides / administration & dosage*
  • Cell-Penetrating Peptides / pharmacology
  • Dendritic Cells / immunology
  • Dendritic Cells / transplantation*
  • Female
  • Forkhead Transcription Factors / antagonists & inhibitors*
  • Humans
  • Immunotherapy
  • Mice
  • T-Lymphocytes, Regulatory / drug effects*
  • T-Lymphocytes, Regulatory / immunology
  • Treatment Outcome
  • Tumor Microenvironment / drug effects
  • Xenograft Model Antitumor Assays

Substances

  • Cancer Vaccines
  • Cell-Penetrating Peptides
  • Forkhead Transcription Factors
  • Foxp3 protein, mouse