The novel preventive effect of Daikenchuto (TJ-100), a Japanese herbal drug, against neonatal necrotizing enterocolitis in rats

Pediatr Surg Int. 2017 Oct;33(10):1109-1114. doi: 10.1007/s00383-017-4145-9. Epub 2017 Aug 16.

Abstract

Purpose: Necrotizing enterocolitis (NEC) is a devastating gastrointestinal disease of premature infants. Daikenchuto, a Japanese herbal drug, has several effects on the digestive system, so we investigated its preventive effects in a rat model of NEC.

Methods: NEC was induced in newborn rats via asphyxia (100% N2 for 90 s; every 4 h) + LPS (4 mg/kg/day [administered orally on days 0 and 1]). The effects of Daikenchuto were evaluated in four groups (control: 0 g/kg/day, I: 0.3 g/kg/day, II: 0.6 g/kg/day, and III: 1.0 g/kg/day). Daikenchuto was administered into the stomach through a microcatheter. The incidence and severity of NEC were pathologically assessed using the NEC grade in accordance with Dovorak's previous report. Cell positivity for inflammatory cytokine (IL-6) was also evaluated.

Results: Daikenchuto reduced the incidence of NEC in control, Groups I, II, and III to 68.7, 30.0, 30.7, and 13.3%, respectively. High-dose Daikenchuto significantly improved the incidence of NEC, and the rate of IL-6 positive cells in group III was significantly lower than in the control group (p = 0.04).

Conclusion: We evaluated the effect of Daikenchuto against NEC and found that it reduced the incidence rate of NEC due to a decrease in the IL-6 production.

Keywords: Daikenchuto; IL-6; NEC grade; Necrotizing enterocolitis; Rat model.

MeSH terms

  • Animals
  • Animals, Newborn
  • Disease Models, Animal
  • Enterocolitis, Necrotizing / prevention & control*
  • Humans
  • Ileum / drug effects
  • Ileum / metabolism
  • Incidence
  • Interleukin-6 / metabolism
  • Panax
  • Plant Extracts / therapeutic use*
  • Rats
  • Rats, Sprague-Dawley
  • Zanthoxylum
  • Zingiberaceae

Substances

  • Interleukin-6
  • Plant Extracts
  • dai-kenchu-to