Tumor-associated B-cells induce tumor heterogeneity and therapy resistance

Nat Commun. 2017 Sep 19;8(1):607. doi: 10.1038/s41467-017-00452-4.

Abstract

In melanoma, therapies with inhibitors to oncogenic BRAFV600E are highly effective but responses are often short-lived due to the emergence of drug-resistant tumor subpopulations. We describe here a mechanism of acquired drug resistance through the tumor microenvironment, which is mediated by human tumor-associated B cells. Human melanoma cells constitutively produce the growth factor FGF-2, which activates tumor-infiltrating B cells to produce the growth factor IGF-1. B-cell-derived IGF-1 is critical for resistance of melanomas to BRAF and MEK inhibitors due to emergence of heterogeneous subpopulations and activation of FGFR-3. Consistently, resistance of melanomas to BRAF and/or MEK inhibitors is associated with increased CD20 and IGF-1 transcript levels in tumors and IGF-1 expression in tumor-associated B cells. Furthermore, first clinical data from a pilot trial in therapy-resistant metastatic melanoma patients show anti-tumor activity through B-cell depletion by anti-CD20 antibody. Our findings establish a mechanism of acquired therapy resistance through tumor-associated B cells with important clinical implications.Resistance to BRAFV600E inhibitors often occurs in melanoma patients. Here, the authors describe a potential mechanism of acquired drug resistance mediated by tumor-associated B cells-derived IGF-1.

Publication types

  • Clinical Trial, Phase II
  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Antibodies, Monoclonal / therapeutic use
  • Antibodies, Monoclonal, Humanized
  • Antineoplastic Agents / therapeutic use*
  • B-Lymphocytes / metabolism*
  • Cell Survival
  • Cisplatin / therapeutic use
  • Drug Resistance, Neoplasm*
  • Fibroblast Growth Factor 2 / metabolism
  • Humans
  • In Vitro Techniques
  • Insulin-Like Growth Factor I / metabolism*
  • Lymphocytes, Tumor-Infiltrating / metabolism*
  • Melanoma / drug therapy*
  • Melanoma / genetics
  • Paclitaxel / therapeutic use
  • Pilot Projects
  • Protein Kinase Inhibitors / therapeutic use*
  • Proto-Oncogene Proteins B-raf / genetics
  • Receptor, Fibroblast Growth Factor, Type 3 / metabolism
  • Skin Neoplasms / drug therapy*
  • Skin Neoplasms / genetics
  • Tumor Microenvironment

Substances

  • Antibodies, Monoclonal
  • Antibodies, Monoclonal, Humanized
  • Antineoplastic Agents
  • IGF1 protein, human
  • Protein Kinase Inhibitors
  • Fibroblast Growth Factor 2
  • Insulin-Like Growth Factor I
  • FGFR3 protein, human
  • Receptor, Fibroblast Growth Factor, Type 3
  • BRAF protein, human
  • Proto-Oncogene Proteins B-raf
  • ofatumumab
  • Paclitaxel
  • Cisplatin