Small Molecules Drive Big Improvements in Immuno-Oncology Therapies

Angew Chem Int Ed Engl. 2018 Apr 9;57(16):4412-4428. doi: 10.1002/anie.201707816. Epub 2018 Feb 22.

Abstract

Immuno-oncology therapies have the potential to revolutionize the armamentarium of available cancer treatments. To further improve clinical response rates, researchers are looking for novel combination regimens, with checkpoint blockade being used as a backbone of the treatment. This Review highlights the significance of small molecules in this approach, which holds promise to provide increased benefit to cancer patients.

Keywords: T-cells; checkpoint inhibitor; combination therapy; kinase inhibitors; small molecules.

Publication types

  • Review

MeSH terms

  • Antineoplastic Agents / chemistry*
  • Antineoplastic Agents / therapeutic use*
  • Humans
  • Immunotherapy*
  • Neoplasms / immunology*
  • Neoplasms / pathology
  • Neoplasms / therapy*
  • Small Molecule Libraries / chemistry*
  • Small Molecule Libraries / therapeutic use*

Substances

  • Antineoplastic Agents
  • Small Molecule Libraries