Kinetic mechanism for the intestinal absorption of ofloxacin

J Pharm Pharmacol. 1988 Mar;40(3):211-2. doi: 10.1111/j.2042-7158.1988.tb05223.x.

Abstract

The absorptive behaviour of ofloxacin, a quinolone antibacterial agent, was studied following recirculation in small intestine of both male and female rats, at initial doses ranging from 0.125 to 5 mg mL-1. A saturable Michaelis-Menten process is suggested to explain the intestinal absorption. No significant differences were found in the absorption parameters per metabolic weight unit.

MeSH terms

  • Animals
  • Anti-Infective Agents / pharmacokinetics*
  • Chromatography, High Pressure Liquid
  • Female
  • In Vitro Techniques
  • Intestinal Absorption*
  • Male
  • Ofloxacin
  • Oxazines / pharmacokinetics*
  • Perfusion
  • Rats
  • Rats, Inbred Strains

Substances

  • Anti-Infective Agents
  • Oxazines
  • Ofloxacin