Improved Pulse Wave Velocity and Renal Function in Individualized Calcineurin Inhibitor Treatment by Immunomonitoring: The Randomized Controlled Calcineurin Inhibitor-Sparing Trial

Transplantation. 2018 Mar;102(3):510-520. doi: 10.1097/TP.0000000000001973.

Abstract

Background: A new immune monitoring tool which assesses the expression of nuclear factor of activated T cells (NFAT)-regulated genes measures the functional effects of cyclosporine A. This is the first prospective randomized controlled study to compare standard pharmacokinetic monitoring by cyclosporine trough levels to NFAT-regulated gene expression (NFAT-RE).

Methods: Expression of the NFAT-regulated genes was determined by qRT-PCR at cyclosporine trough and peak level. Cardiovascular risk was assessed by change of pulse wave velocity from baseline to month 6. Clinical follow-up was 12 months.

Results: In total, 55 stable kidney allograft recipients were enrolled. Mean baseline residual NFAT-RE was 13.1 ± 9.1%. Patients in the NFAT-RE group showed a significant decline in pulse wave velocity from baseline to month 6 versus the standard group (-1.7 ± 2.0 m/s vs 0.4 ± 1.4 m/s, P < 0.001). Infections occurred more often in the standard group compared with the immune monitoring group. No opportunistic infections occurred with NFAT-RE monitoring. At 12 months of follow-up, renal function was significantly better with NFAT-RE versus standard monitoring (Nankivell glomerular filtration rate: 68.5 ± 17.4 mL/min vs 57.2 ± 19.0 mL/min; P = 0.009).

Conclusions: NFAT-RE as translational immune monitoring tool proved efficacious and safe in individualizing cyclosporine therapy, with the opportunity to reduce the cardiovascular risk and improve long-term renal allograft function.

Publication types

  • Randomized Controlled Trial
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Calcineurin Inhibitors / adverse effects
  • Calcineurin Inhibitors / pharmacology*
  • Cardiovascular Diseases / etiology
  • Cyclosporine / pharmacology
  • Glomerular Filtration Rate / drug effects*
  • Humans
  • Kidney Transplantation*
  • NFATC Transcription Factors / genetics
  • Prospective Studies
  • Pulse Wave Analysis*

Substances

  • Calcineurin Inhibitors
  • NFATC Transcription Factors
  • Cyclosporine

Associated data

  • ISRCTN/ISRCTN3222
  • EudraCT/2011-003547-21