Four new monacolin analogs from Monascus purpureus-fermented rice

J Asian Nat Prod Res. 2018 Mar;20(3):209-216. doi: 10.1080/10286020.2017.1396978. Epub 2017 Nov 8.

Abstract

Four new monacolin analogs, monacolin T (1), monacolin U (2) 6a-O-methyl-4,6-dihydromonacolin L (3), and 6a-O-ethyl-4,6-dihydromonacolin L (4) were isolated from the ethanolic extract of Monascus purpureus-fermented rice. Their structures were determined by a combination of 1D, 2D NMR experiments (1H-1HCOSY, HSQC, HMBC, and ROESY), and mass spectrometry. In vitro cytotoxic assay, all compounds were inactive at the concentration of 10 µM.

Keywords: Monascus purpureus; isolation and elucidation; monacolin analogs.

MeSH terms

  • Drug Screening Assays, Antitumor
  • Fermentation
  • Molecular Structure
  • Monascus / chemistry*
  • Naphthalenes / chemistry
  • Naphthalenes / isolation & purification*
  • Oryza / microbiology*

Substances

  • Naphthalenes
  • monacolin T