Structural basis of cholesterol binding by a novel clade of dendritic cell modulators from ticks

Sci Rep. 2017 Nov 22;7(1):16057. doi: 10.1038/s41598-017-16413-2.

Abstract

Two crystal structures of Japanin, an 18 kDa immune-modulatory lipocalin from the Brown Ear Tick (Rhipicephalus appendiculatus), have been determined at 2.2 and 2.4 Å resolution. In both crystal forms the protein is in complex with cholesterol, which sits in a closed pocket at the centre of the lipocalin barrel. Both crystal forms are dimers, which are also observed in solution. Molecular modelling suggests that previously-described members of a tick protein family bearing high sequence homology to Japanin are also likely to bind cholesterol or cholesterol derivatives.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Amino Acid Sequence
  • Animals
  • Binding Sites
  • Cholesterol / metabolism*
  • Crystallography, X-Ray
  • Dendritic Cells / metabolism*
  • Dimerization
  • Lipocalins / chemistry
  • Lipocalins / metabolism
  • Protein Structure, Secondary
  • Rhipicephalus / metabolism*
  • Structural Homology, Protein

Substances

  • Lipocalins
  • Cholesterol