The diverse functions of the hepatitis B core/capsid protein (HBc) in the viral life cycle: Implications for the development of HBc-targeting antivirals

Antiviral Res. 2018 Jan:149:211-220. doi: 10.1016/j.antiviral.2017.11.015. Epub 2017 Nov 26.

Abstract

Virally encoded proteins have evolved to perform multiple functions, and the core protein (HBc) of the hepatitis B virus (HBV) is a perfect example. While HBc is the structural component of the viral nucleocapsid, additional novel functions for the nucleus-localized HBc have recently been described. These results extend for HBc, beyond its structural role, a regulatory function in the viral life cycle and potentially a role in pathogenesis. In this article, we review the diverse roles of HBc in HBV replication and pathogenesis, emphasizing how the unique structure of this protein is key to its various functions. We focus in particular on recent advances in understanding the significance of HBc phosphorylations, its interaction with host proteins and the role of HBc in regulating the transcription of host genes. We also briefly allude to the emerging niche for new direct-acting antivirals targeting HBc, known as Core (protein) Allosteric Modulators (CAMs).

Keywords: CAMs; Core allosteric modulators; HBV; HBV core antigen; HBc; HBc phosphorylations; HBc structure; Hepatitis B virus; PLK1.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't
  • Review

MeSH terms

  • Animals
  • Antiviral Agents / pharmacology
  • Antiviral Agents / therapeutic use
  • Drug Discovery
  • Gene Expression Regulation, Viral
  • Hepatitis B / drug therapy
  • Hepatitis B / virology*
  • Hepatitis B Core Antigens / chemistry
  • Hepatitis B Core Antigens / genetics
  • Hepatitis B Core Antigens / metabolism*
  • Hepatitis B virus / drug effects
  • Hepatitis B virus / physiology*
  • Host-Pathogen Interactions
  • Humans
  • Phosphorylation
  • Protein Binding
  • Protein Transport
  • Viral Core Proteins / antagonists & inhibitors
  • Viral Core Proteins / chemistry
  • Viral Core Proteins / genetics
  • Viral Core Proteins / metabolism*

Substances

  • Antiviral Agents
  • Hepatitis B Core Antigens
  • Viral Core Proteins