Bioaccessibility, cellular uptake and transport of luteins and assessment of their antioxidant activities

Food Chem. 2018 May 30:249:66-76. doi: 10.1016/j.foodchem.2017.12.055. Epub 2017 Dec 14.

Abstract

A rapid method for producing 9Z- and 13'Z-isomers from all-E-lutein was developed using I-TiO2 as catalyst. In a simulated in vitro gastrointestinal digestion model, both trans-cis isomerization of all-E-lutein and cis-trans isomerization of Z-luteins occurred during the intestinal phase. The bioaccessibility of all isomers was between 14 and 23%, and it was higher for Z-luteins. In a Caco-2 cell monolayer model, all isomers were relatively stable during cellular uptake and transport across the membrane as no significant isomerization and degradation was detected, but all-E-lutein exhibited significantly higher cellular uptake and transport efficiencies. These results suggest that Z-luteins found in human plasma may likely be formed before intestinal absorption. 13'Z-Lutein also exhibited highest antioxidant activity in FRAP, DPPH and ORAC-L assays, but no significant difference in cell-based antioxidant assay compared with other isomers. Future studies on the different antioxidant activities of cis isomers of lutein in vivo will provide further explanation.

Keywords: Antioxidant activity; Bioaccessibility; Caco-2 cells; Cellular uptake; Isomerization; Lutein; cis-Isomers.

MeSH terms

  • Antioxidants / chemistry
  • Antioxidants / pharmacology*
  • Biological Transport
  • Caco-2 Cells
  • Digestion
  • Humans
  • Intestinal Absorption
  • Isomerism
  • Lutein / chemistry
  • Lutein / metabolism
  • Lutein / pharmacokinetics*
  • Lutein / pharmacology

Substances

  • Antioxidants
  • Lutein