Vascular niche IL-6 induces alternative macrophage activation in glioblastoma through HIF-2α

Nat Commun. 2018 Feb 8;9(1):559. doi: 10.1038/s41467-018-03050-0.

Abstract

Spatiotemporal regulation of tumor immunity remains largely unexplored. Here we identify a vascular niche that controls alternative macrophage activation in glioblastoma (GBM). We show that tumor-promoting macrophages are spatially proximate to GBM-associated endothelial cells (ECs), permissive for angiocrine-induced macrophage polarization. We identify ECs as one of the major sources for interleukin-6 (IL-6) expression in GBM microenvironment. Furthermore, we reveal that colony-stimulating factor-1 and angiocrine IL-6 induce robust arginase-1 expression and macrophage alternative activation, mediated through peroxisome proliferator-activated receptor-γ-dependent transcriptional activation of hypoxia-inducible factor-2α. Finally, utilizing a genetic murine GBM model, we show that EC-specific knockout of IL-6 inhibits macrophage alternative activation and improves survival in the GBM-bearing mice. These findings illustrate a vascular niche-dependent mechanism for alternative macrophage activation and cancer progression, and suggest that targeting endothelial IL-6 may offer a selective and efficient therapeutic strategy for GBM, and possibly other solid malignant tumors.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Arginase / immunology
  • Basic Helix-Loop-Helix Transcription Factors / genetics*
  • Cell Line, Tumor
  • Cells, Cultured
  • Disease Progression
  • Endothelial Cells / immunology*
  • Glioblastoma / immunology*
  • Humans
  • Interleukin-6 / immunology*
  • Macrophage Activation / immunology*
  • Macrophage Colony-Stimulating Factor / immunology
  • Macrophages / immunology*
  • Mice
  • Microvessels / cytology
  • Monocytes / immunology
  • Neoplasms, Experimental / immunology
  • Transcriptional Activation
  • Tumor Microenvironment

Substances

  • Basic Helix-Loop-Helix Transcription Factors
  • Interleukin-6
  • endothelial PAS domain-containing protein 1
  • Macrophage Colony-Stimulating Factor
  • ARG1 protein, human
  • Arg1 protein, mouse
  • Arginase